SCHEMBL28622149

SCHEMBL28622149

Clc1ccc2nc(-c3ccccc3)cc(Cc3ccccc3)c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.56
DHODH Q02127 6/20 0.53
AURKA O14965 1/20 0.51
AURKB Q96GD4 1/20 0.51
HPGD P15428 3/20 0.47
ALDH1A1 P00352 2/20 0.47
HIF1A Q16665 2/20 0.47
HSD17B10 Q99714 2/20 0.47
PTGES O14684 1/20 0.47
ALOX5 P09917 1/20 0.47
CYP2C9 P11712 1/20 0.47
CASP7 P55210 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MEN1 O00255 1/20 0.46
CYP3A4 P08684 1/20 0.46
ALOX15 P16050 1/20 0.46
KMT2A Q03164 1/20 0.46
ELANE P08246 1/20 0.44
KDM4E B2RXH2 2/20 0.44
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28619856 0.84 ACHE (0.56) DHODHHPGDCYP2C9SMN1; SMN2KDM4E
SCHEMBL28634603 0.84 DHODH (0.54) MAPK1DHODHHPGDPTGESSMN1; SMN2
SCHEMBL28623574 0.82 DHODH (0.54) DHODHALDH1A1MEN1KMT2AMAPT
SCHEMBL28626532 0.82 DHODH (0.60) MAPK1DHODHHPGDALDH1A1HSD17B10
SCHEMBL28626601 0.79 KDM4E (0.64) DHODHAURKAAURKBHPGDALDH1A1
SCHEMBL8956330 0.78 MAPK1 (0.85) MAPK1DHODHAURKAAURKBHPGD
SCHEMBL10864591 0.78 MAPK1 (0.65) MAPK1DHODHAURKAAURKBHPGD
SCHEMBL8410911 0.76 MAPK1 (0.82) MAPK1DHODHAURKAAURKBHPGD
SCHEMBL10609537 0.75 MAPK1 (0.61) MAPK1DHODHAURKAAURKBHPGD
SCHEMBL16098232 0.75 MAPK1 (0.54) MAPK1DHODHAURKAAURKBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113277978-B Preparation method of 2, 4-disubstituted quinoline compound 河南师范大学 2022-06-03 CN disclosed
CN-113277978-A Preparation method of 2, 4-disubstituted quinoline compound 河南师范大学 2021-08-20 CN disclosed