SCHEMBL2862276

SCHEMBL2862276

Cc1cccc(CNC(=O)c2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)c1

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 14/20 0.70
HSP90AA1 P07900 1/20 0.54
MAPT P10636 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
TRPC3 Q13507 1/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HPGD P15428 1/20 0.49
DDT P30046 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2861171 0.91 CCR1 (0.69) CCR1NPSR1KDM4EALDH1A1HPGD
SCHEMBL2860538 0.91 KDM4E (0.61) CCR1MAPTKDM4EALDH1A1HPGD
SCHEMBL2859933 0.89 CCR1 (0.80) CCR1HSP90AA1MAPTNPSR1HPGD
SCHEMBL2852015 0.88 CCR1 (0.63) CCR1HSP90AA1MAPTNPSR1TRPC3
SCHEMBL2854508 0.85 CCR1 (0.62) CCR1HSP90AA1MAPTNPSR1KDM4E
SCHEMBL2854425 0.85 CCR1 (0.60) CCR1MAPTTRPC3KDM4EALDH1A1
SCHEMBL2854543 0.84 CCR1 (0.54) CCR1HSP90AA1MAPTNPSR1DDT
SCHEMBL2855565 0.84 CCR1 (0.66) CCR1HSP90AA1MAPTNPSR1TRPC3
SCHEMBL2855315 0.83 KDM4E (0.65) CCR1MAPTKDM4EALDH1A1HPGD
SCHEMBL2852818 0.83 NPC1 (0.50) CCR1MAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed