SCHEMBL2854508

SCHEMBL2854508

O=C(NCc1cccc([N+](=O)[O-])c1)c1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 15/20 0.62
AKR1B1 P15121 1/20 0.53
ACHE P22303 1/20 0.51
HSP90AA1 P07900 1/20 0.49
MAPT P10636 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2852816 0.89 ACHE (0.59) CCR1ACHEMAPTNPSR1KDM4E
SCHEMBL2858942 0.86 CCR1 (0.82) CCR1ACHEHSP90AA1MAPTNPSR1
SCHEMBL2859933 0.86 CCR1 (0.80) CCR1HSP90AA1MAPTNPSR1
SCHEMBL2856514 0.85 CCR1 (0.49) CCR1AKR1B1ACHEHSP90AA1MAPT
SCHEMBL2862276 0.85 CCR1 (0.70) CCR1HSP90AA1MAPTNPSR1KDM4E
SCHEMBL2855062 0.85 CCR1 (0.65) CCR1ACHEMAPTNPSR1KDM4E
SCHEMBL2852015 0.84 CCR1 (0.63) CCR1HSP90AA1MAPTNPSR1KDM4E
SCHEMBL2860444 0.84 CCR1 (0.60) CCR1ACHEMAPTNPSR1KDM4E
SCHEMBL2854425 0.82 CCR1 (0.60) CCR1MAPTKDM4EALDH1A1
SCHEMBL2852112 0.81 CCR1 (0.68) CCR1ACHEMAPTNPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed