SCHEMBL28624312

SCHEMBL28624312

CNC(=O)NC1CCN(C(=O)[C@@H](CCCCNC(N)=O)OC(=O)NCc2ccccc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.45
MEN1 O00255 1/20 0.44
POLB P06746 1/20 0.44
KMT2A Q03164 1/20 0.44
DRD4 P21917 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
KDM5A P29375 1/20 0.40
RAB9A P51151 1/20 0.40
EPHX1 P07099 2/20 0.39
HPGD P15428 1/20 0.39
KEAP1 Q14145 2/20 0.38
NFE2L2 Q16236 2/20 0.38
F13A1 P00488 1/20 0.38
TGM2 P21980 1/20 0.38
TGM1 P22735 1/20 0.38
TSHR P16473 1/20 0.37
TPSAB1 Q15661 1/20 0.37
SMYD3 Q9H7B4 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28611634 0.91 MAPT (0.44) MAPTMEN1POLBKMT2ADRD4
Hydrochloric Acid SCHEMBL28613881 0.90 MAPT (0.44) MAPTMEN1POLBKMT2ADRD4
SCHEMBL28624314 0.81 TGM2 (0.59) F13A1TGM2TGM1
SCHEMBL28625098 0.79 EPHX2 (0.44) EPHX1
SCHEMBL28613203 0.75 EPHX2 (0.44) KDM5AEPHX1
SCHEMBL28613201 0.75 EPHX2 (0.44) KDM5AEPHX1
SCHEMBL21738934 0.72 OPRK1 (0.64)
SCHEMBL28613211 0.71 EPHX2 (0.35) KDM5AEPHX1TSHRTPSAB1
SCHEMBL28613209 0.71 EPHX2 (0.35) KDM5AEPHX1TSHRTPSAB1
SCHEMBL28624310 0.69 EPHX2 (0.48) EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107098871-B Phenyl propionamide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-07-02 CN disclosed