SCHEMBL28625910

SCHEMBL28625910

CC1CCN(Cc2ccc3nc(NC(=O)c4cc5cccc(O)c5oc4=O)sc3c2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.51
TP53 P04637 2/20 0.44
LMNA P02545 1/20 0.44
HCAR1 Q9BXC0 2/20 0.44
HSD17B1 P14061 1/20 0.44
HSD17B2 P37059 1/20 0.44
PCSK9 Q8NBP7 2/20 0.43
SSTR5 P35346 2/20 0.42
MAPT P10636 1/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ESR1 P03372 1/20 0.41
POLB P06746 1/20 0.41
PKM P14618 1/20 0.41
HPGD P15428 1/20 0.41
CACNA1B Q00975 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28629444 0.93 CASP3 (0.53) CASP3HCAR1HSD17B1HSD17B2PCSK9
SCHEMBL28630602 0.91 HPGD (0.53) CASP3TP53SSTR5MAPTMEN1
SCHEMBL28621580 0.85 ALDH1A1 (0.52) CASP3TP53HCAR1SSTR5MAPT
SCHEMBL28636610 0.83 AKR1C3 (0.52) TP53MAPTMEN1KMT2AALDH1A1
SCHEMBL28626050 0.81 HSD17B1 (0.49) CASP3TP53LMNAHSD17B1HSD17B2
SCHEMBL28621873 0.80 HSD17B1 (0.48) CASP3TP53LMNAHSD17B1HSD17B2
SCHEMBL28621577 0.78 POLB (0.46) TP53MAPTMEN1KMT2AALDH1A1
SCHEMBL28621589 0.76 CASP3 (0.56) CASP3LMNAHCAR1PCSK9NPC1
SCHEMBL28621593 0.75 AKR1B10 (0.44) CASP3HSD17B1HSD17B2PCSK9MAPT
SCHEMBL28641065 0.73 TP53 (0.67) TP53MAPTRAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108715589-B Coumarin derivative used as caspase-3 activator and application thereof 华侨大学 2021-04-20 CN disclosed