SCHEMBL2862872

SCHEMBL2862872

Cc1nn(C)c(C)c1OC(=O)NCc1cccc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 5/20 0.47
KDM4E B2RXH2 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
FAAH O00519 1/20 0.46
THRB P10828 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MLYCD O95822 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
PLA2G1B P04054 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
GAA P10253 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
ATG4B Q9Y4P1 1/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2859060 0.89 ALDH1A1 (0.46) KDM4ENPSR1MLYCDCYP1A2CYP3A4
SCHEMBL2861199 0.83 AOC3 (0.49)
SCHEMBL2857918 0.81 CCR1 (0.54) CCR1MLYCDNPC1KMT2AMEN1
SCHEMBL2854621 0.78 TSHR (0.58) NPC1RAB9AKMT2AMEN1TSHR
SCHEMBL2854535 0.74 SMN1; SMN2 (0.60) L3MBTL1NPC1RAB9AKMT2AMEN1
SCHEMBL24713417 0.74 MAPK14 (0.66) KDM4EFAAHL3MBTL1MLYCDKMT2A
SCHEMBL2857889 0.74 NPC1 (0.52) NPC1RAB9AKMT2AGAA
SCHEMBL24713418 0.74 USP2 (0.62) KDM4EFAAHMLYCDNPC1RAB9A
SCHEMBL2854225 0.73 CCR1 (0.60) CCR1KDM4ENPSR1MAPK14
SCHEMBL24713109 0.73 MLYCD (0.67) KDM4ENPSR1L3MBTL1MLYCDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed