SCHEMBL28629610

SCHEMBL28629610

O=C(O)CCC(=O)c1cc(F)cc(I)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.46
ALDH1A1 P00352 3/20 0.42
CYP2C19 P33261 2/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP1A2 P05177 3/20 0.41
RAB9A P51151 2/20 0.41
FFAR1 O14842 1/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HIF1A Q16665 1/20 0.41
USP5 P45974 1/20 0.39
PKM P14618 1/20 0.38
TSHR P16473 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
HCAR1 Q9BXC0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29399457 1.00 NR4A2 (0.46) NR4A2ALDH1A1CYP2C19GAAKMT2A
SCHEMBL5081101 0.87 NR4A2 (0.54) NR4A2ALDH1A1CYP2C19GAAKMT2A
SCHEMBL22097301 0.79 KMT2A (0.55) NR4A2ALDH1A1CYP2C19GAAKMT2A
SCHEMBL1947967 0.77 HCAR1 (0.59) ALDH1A1LMNASMN1; SMN2HIF1ATSHR
SCHEMBL5080184 0.76 HDAC3 (0.55) NR4A2RAB9ALMNATSHRL3MBTL1
SCHEMBL30416829 0.75 ALDH1A1 (0.55) NR4A2ALDH1A1CYP2C19KMT2ACYP1A2
SCHEMBL20703168 0.73 CES2 (0.52) NR4A2ALDH1A1CYP2C19GAAKMT2A
SCHEMBL2691520 0.73 NR4A2 (0.62) NR4A2ALDH1A1CYP2C19GAAKMT2A
SCHEMBL21516794 0.72 PARP1 (0.52) CYP2C19CYP1A2SMN1; SMN2TSHRL3MBTL1
SCHEMBL31585604 0.71 HCAR2 (0.61) NR4A2ALDH1A1CYP2C19GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109608464-B Radioiodine-labeled Larotrectinib compound and preparation method and application thereof 上海健康医学院 2021-09-24 CN claimed
CN-109608464-B Radioiodine-labeled Larotrectinib compound and preparation method and application thereof 上海健康医学院 2021-09-24 CN disclosed