SCHEMBL2856121

SCHEMBL2856121

Cc1cnc(N2CCC(NC(=O)C#CC(=O)c3ccccc3C)C2)s1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 1/20 0.40
BTK Q06187 2/20 0.37
HRH3 Q9Y5N1 1/20 0.37
ACKR3 P25106 3/20 0.36
AKT1 P31749 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
POLB P06746 1/20 0.36
CHRNA7 P36544 2/20 0.35
HTR7 P34969 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 1/20 0.35
DPP4 P27487 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL973571 0.85 HRH3 (0.37) PAK1BTKHRH3ACKR3AKT1
SCHEMBL2861257 0.85 SMN1; SMN2 (0.37) PAK1BTKACKR3MEN1KMT2A
SCHEMBL2856320 0.84 CHRNA7 (0.40) PAK1BTKHRH3ACKR3KMT2A
SCHEMBL973764 0.83 BTK (0.45) BTKHRH3ACKR3AKT1CHRNA7
SCHEMBL2862996 0.83 CCNE1 (0.38) BTKHRH3ACKR3MEN1KMT2A
SCHEMBL2855060 0.83 ALDH1A1 (0.43) PAK1BTKHRH3ACKR3MEN1
SCHEMBL972148 0.81 GRM5 (0.39) BTKHRH3ACKR3MEN1KMT2A
SCHEMBL975872 0.80 CA12 (0.41) BTKHRH3ACKR3CHRNA7ALDH1A1
SCHEMBL2854730 0.80 CTSB (0.37) PAK1BTKACKR3MEN1KMT2A
SCHEMBL974821 0.79 HRH3 (0.38) PAK1BTKHRH3ACKR3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968957-B1 SUBSTITUTED THIAZOLES AND THEIR USE FOR PRODUCING DRUGS GRUENENTHAL GMBH (DE) 2010-01-20 EP claimed