SCHEMBL2856320

SCHEMBL2856320

Cc1ccc(C(=O)C#CC(=O)NC2CCN(c3ncc(C)s3)C2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.40
PAK1 Q13153 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
BTK Q06187 1/20 0.36
KARS1 Q15046 1/20 0.36
DPP4 P27487 1/20 0.36
ACKR3 P25106 2/20 0.36
TMPRSS15 P98073 2/20 0.35
SMPD3 Q9NY59 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2862996 0.89 CCNE1 (0.38) CHRNA7HRH3BTKACKR3CCNE1
SCHEMBL974821 0.87 HRH3 (0.38) CHRNA7PAK1HRH3BTKDPP4
SCHEMBL2856121 0.84 PAK1 (0.40) CHRNA7PAK1HRH3BTKDPP4
SCHEMBL2863170 0.84 PPARG (0.36) PAK1BTKKARS1DPP4SMPD3
SCHEMBL2854222 0.82 SMN1; SMN2 (0.40) PAK1HRH3BTKKARS1DPP4
SCHEMBL973764 0.81 BTK (0.45) CHRNA7HRH3BTKDPP4ACKR3
SCHEMBL973812 0.80 HRH3 (0.38) CHRNA7HRH3BTKDPP4ACKR3
SCHEMBL975864 0.80 BTK (0.38) CHRNA7HRH3BTKACKR3SMPD3
SCHEMBL2853786 0.80 LMNA (0.38) PAK1BTKACKR3KMT2A
SCHEMBL974669 0.79 HRH3 (0.39) CHRNA7HRH3BTKACKR3SMPD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968957-B1 SUBSTITUTED THIAZOLES AND THEIR USE FOR PRODUCING DRUGS GRUENENTHAL GMBH (DE) 2010-01-20 EP claimed