SCHEMBL28633468

SCHEMBL28633468

CCOc1cc2c(cc1Br)CN(Cc1ccccc1)C2=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
HDAC4 P56524 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
LMNA P02545 2/20 0.46
TSHR P16473 1/20 0.46
HTT P42858 1/20 0.46
CASP3 P42574 1/20 0.41
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GRM2 Q14416 1/20 0.40
DHPS P49366 1/20 0.40
MAPT P10636 2/20 0.39
POLB P06746 1/20 0.39
PARP1 P09874 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
IDH1 O75874 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28638401 0.89 HDAC4 (0.48) KMT2AMEN1HDAC4HDAC1HDAC6
SCHEMBL30604584 0.88 GRM5 (0.52) KMT2AMEN1LMNATSHRHTT
SCHEMBL28638924 0.88 GRM5 (0.52) KMT2AMEN1LMNATSHRHTT
SCHEMBL28633462 0.87 KMT2A (0.53) KMT2AMEN1HDAC4HDAC1HDAC6
SCHEMBL28639031 0.82 KMT2A (0.57) KMT2AMEN1HDAC4HDAC1HDAC6
SCHEMBL29630709 0.81 ACHE (0.48) HDAC4HDAC1HDAC6KDM4EDRD4
SCHEMBL28643695 0.79 LRRK2 (0.37) HDAC4HDAC1HDAC6LMNATSHR
SCHEMBL24823388 0.78 HDAC1 (0.50) KMT2AMEN1HDAC4HDAC1HDAC6
SCHEMBL28656932 0.78 HDAC1 (0.53) KMT2AMEN1HDAC4HDAC1HDAC6
SCHEMBL28641201 0.77 GRM5 (0.58) KMT2AMEN1LMNADHPSDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493438-B Tetrahydroisoquinoline compounds 南京再明医药有限公司 2023-10-20 CN disclosed
CN-113493438-A Tetrahydroisoquinoline compounds 江苏先声药业有限公司 2021-10-12 CN disclosed