SCHEMBL28633752

SCHEMBL28633752

O=c1[nH]c(-c2nc3ccccc3[nH]2)cc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.56
FGFR1 P11362 6/20 0.56
PDGFRB P09619 5/20 0.56
NPC1 O15118 5/20 0.53
RAB9A P51151 4/20 0.53
KDM4E B2RXH2 2/20 0.53
ALDH1A1 P00352 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
ABCB11 O95342 1/20 0.53
TP53 P04637 1/20 0.53
PKM P14618 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
HSD17B10 Q99714 1/20 0.53
AURKA O14965 1/20 0.53
CDK1 P06493 1/20 0.53
CDK2 P24941 1/20 0.53
AURKB Q96GD4 1/20 0.53
FLT1 P17948 3/20 0.52
CHEK1 O14757 2/20 0.52
LMNA P02545 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4497587 0.82 TNKS (0.59) KDRFGFR1PDGFRBNPC1RAB9A
SCHEMBL924438 0.80 ESR1 (0.71) KDRFGFR1PDGFRBNPC1RAB9A
SCHEMBL27635441 0.80 KDM4E (0.57) KDRFGFR1PDGFRBNPC1RAB9A
SCHEMBL27824964 0.76 ALDH1A1 (0.62) KDRFGFR1PDGFRBNPC1RAB9A
SCHEMBL21297858 0.74 HPGD (0.63) KDRFGFR1PDGFRBNPC1RAB9A
SCHEMBL7256021 0.72 ESR1 (0.54) KDRFGFR1PDGFRBNPC1RAB9A
SCHEMBL30305373 0.72 KDR (0.78) KDRFGFR1PDGFRBNPC1RAB9A
SCHEMBL3503147 0.72 KDR (1.00) KDRFGFR1PDGFRBNPC1RAB9A
SCHEMBL30561047 0.72 NPC1 (1.00) NPC1RAB9AKDM4EALDH1A1SMN1; SMN2
SCHEMBL172216 0.72 NPC1 (1.00) NPC1RAB9AKDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114181214-A Non-activated alkane C (sp)3) -H-functional initiated radical cyclization reaction process 宁波大学 2022-03-15 CN claimed
CN-113373465-B Method for synthesizing silicon-based substituted benzimidazolo isoquinolinone compounds through photoelectric concerted catalysis 北京工业大学 2022-06-14 CN disclosed
CN-114181214-A Non-activated alkane C (sp)3) -H-functional initiated radical cyclization reaction process 宁波大学 2022-03-15 CN disclosed
CN-114181214-A Non-activated alkane C (sp)3) -H-functional initiated radical cyclization reaction process 宁波大学 2022-03-15 CN disclosed
CN-113980016-A Method for preparing benzimidazol isoquinolinone compound 怀化学院 2022-01-28 CN disclosed
CN-113373465-A Method for synthesizing silicon-based substituted benzimidazolo isoquinolinone compounds through photoelectric concerted catalysis 北京工业大学 2021-09-10 CN disclosed