SCHEMBL28634835

SCHEMBL28634835

CCn1c(N)c(NC(=O)/C=C/c2ccc(Br)cc2)c(=O)n(CC)c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.45
LMNA P02545 5/20 0.42
RAB9A P51151 2/20 0.42
KDM4E B2RXH2 2/20 0.42
GPR183 P32249 1/20 0.41
TRPA1 O75762 1/20 0.41
TRPM8 Q7Z2W7 1/20 0.41
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MAPT P10636 2/20 0.39
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
THRB P10828 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
ALDH1A1 P00352 2/20 0.38
TRPV1 Q8NER1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28627469 0.87 SLC6A19 (0.53) MCHR1RAB9AKDM4EHDAC1HDAC8
SCHEMBL28887209 0.86 ALDH1A1 (0.42) LMNARAB9AKDM4EGPR183HDAC1
SCHEMBL28887208 0.86 ALDH1A1 (0.42) LMNARAB9AKDM4EGPR183HDAC1
SCHEMBL28456104 0.82 SAE1 (0.45) LMNARAB9AKDM4EHDAC1HDAC8
SCHEMBL30632573 0.82 MEN1 (0.52) RAB9AKDM4ESMN1; SMN2NPSR1MAPT
SCHEMBL28515989 0.81 NPC1 (0.48) LMNARAB9AKDM4EHDAC1SMN1; SMN2
SCHEMBL30035914 0.81 NPC1 (0.48) LMNARAB9AKDM4EHDAC1SMN1; SMN2
SCHEMBL28372132 0.80 MAPT (0.39) LMNARAB9AKDM4EHDAC1SMN1; SMN2
SCHEMBL30035241 0.79 VCP (0.38) LMNARAB9AHDAC1SMN1; SMN2NPSR1
SCHEMBL28528919 0.79 HDAC1 (0.36) LMNARAB9AKDM4EHDAC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111072663-B 8-substituted styrylxanthine derivatives and uses thereof 广东东阳光药业有限公司 2021-10-01 CN disclosed
CN-111072663-A 8-substituted styrylxanthine derivatives and uses thereof 广东东阳光药业有限公司 2020-04-28 CN disclosed