SCHEMBL28636765

SCHEMBL28636765

Oc1c(Br)ccc2occc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
HPGD P15428 3/20 0.42
CYP3A4 P08684 2/20 0.42
MAPT P10636 2/20 0.42
CYP2A6 P11509 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KDM4E B2RXH2 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
HSD17B10 Q99714 1/20 0.39
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36
NFKB1 P19838 1/20 0.36
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
FTO Q9C0B1 2/20 0.33
PAX8 Q06710 1/20 0.33
TDP1 Q9NUW8 2/20 0.32
USP2 O75604 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5501432 0.74 POLB (0.42) ALDH1A1HPGDCYP3A4MAPTCYP2A6
SCHEMBL16762286 0.74 MAOA (0.36) CYP2A6MAOAMAOBNFKB1HTR2A
SCHEMBL16048354 0.74 MAOA (0.36) MAOAMAOBNFKB1HTR2AHTR2C
SCHEMBL2048407 0.74 ALDH1A1 (0.42) ALDH1A1HPGDCYP3A4MAPTCYP2A6
SCHEMBL4429415 0.72 PAX8 (0.48) ALDH1A1HPGDCYP3A4MAPTCYP2A6
SCHEMBL4421214 0.72 CYP3A4 (0.68) ALDH1A1HPGDCYP3A4MAPTCYP2A6
SCHEMBL2367986 0.70 TDP1 (0.46) ALDH1A1HPGDCYP3A4MAPTKDM4E
SCHEMBL30382539 0.70 TDP1 (0.46) ALDH1A1HPGDCYP3A4MAPTKDM4E
SCHEMBL11926014 0.69 ALDH1A1 (0.39) ALDH1A1HPGDCYP3A4MAPTCYP2A6
SCHEMBL9079188 0.69 ALDH1A1 (0.42) ALDH1A1HPGDCYP3A4MAPTCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4642784-A1 HETEROCYCLIC AND HETEROARYL COMPOUNDS AS INHIBITORS OF NLRP3 PTC Therapeutics, Inc. (US) 2025-11-05 EP disclosed
WO-2024145623-A1 HETEROCYCLIC AND HETEROARYL COMPOUNDS AS INHIBITORS OF NLRP3 PTC THERAPEUTICS, INC. (US) 2024-07-04 WO disclosed
CN-113087722-B Tricyclic isoxazole compound and preparation method and application thereof 中国人民解放军海军军医大学 2023-04-28 CN disclosed
CN-109438471-B Tricyclic isoxazole compound and preparation method and application thereof 中国人民解放军第二军医大学 2021-09-17 CN disclosed
CN-113087722-A Tricyclic isoxazole compound and preparation method and application thereof 中国人民解放军海军军医大学 2021-07-09 CN disclosed