SCHEMBL28640311

SCHEMBL28640311

COC(=O)C1CCN(Cc2ccccc2)C(C)(C)O1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD17B10 Q99714 1/20 0.43
FKBP1A P62942 1/20 0.42
DRD4 P21917 1/20 0.41
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
CASP1 P29466 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40
SIGMAR1 Q99720 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6819861 0.76 SIGMAR1 (0.49) ALDH1A1SIGMAR1
SCHEMBL21758314 0.75 FKBP1A (0.45) ALDH1A1MAPTHPGDNPSR1HSD17B10
SCHEMBL28878129 0.73 ALDH1A1 (0.43) ALDH1A1MAPTHPGDNPSR1HSD17B10
SCHEMBL21553747 0.72 FKBP1A (0.52) ALDH1A1MAPTHPGDNPSR1HSD17B10
SCHEMBL21553748 0.72 FKBP1A (0.52) ALDH1A1MAPTHPGDNPSR1HSD17B10
SCHEMBL1440209 0.71 ALDH1A1 (0.46) ALDH1A1MAPTHPGDNPSR1HSD17B10
SCHEMBL13657453 0.71 HTR2C (0.46) ALDH1A1MAPTNPSR1FKBP1ACYP3A4
SCHEMBL2069105 0.69 GRIN2B (0.54) DRD4
SCHEMBL12696580 0.69 GRIN2B (0.54) DRD4
SCHEMBL22117717 0.69 NR1H2 (0.52) DRD4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112739698-A Tetrahydropyrimidine derivatives as AHR modulators 捷豹治疗有限公司 2021-04-30 CN disclosed