SCHEMBL28645265

SCHEMBL28645265

COC[C@@H](NCCNC(=O)OCc1ccccc1)C(=O)OC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
HTT P42858 1/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
MAPT P10636 1/20 0.51
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CTSK P43235 2/20 0.48
KYNU Q16719 1/20 0.48
SLC1A3 P43003 1/20 0.47
SLC1A1 P43005 1/20 0.47
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
CTSS P25774 1/20 0.47
TGM2 P21980 1/20 0.47
TRPM8 Q7Z2W7 1/20 0.46
ALDH1A1 P00352 1/20 0.46
ALOX15 P16050 1/20 0.46
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13664696 0.93 HTT (0.56) LMNASMN1; SMN2HTTL3MBTL1MAPT
SCHEMBL344091 0.88 LMNA (0.50) LMNASMN1; SMN2HTTL3MBTL1MAPT
SCHEMBL344090 0.88 LMNA (0.50) LMNASMN1; SMN2HTTL3MBTL1MAPT
SCHEMBL28221031 0.86 LMNA (0.53) LMNASMN1; SMN2HTTL3MBTL1MAPT
SCHEMBL28221007 0.83 LMNA (0.58) LMNASMN1; SMN2HTTL3MBTL1MAPT
SCHEMBL28221005 0.83 LMNA (0.58) LMNASMN1; SMN2HTTL3MBTL1MAPT
SCHEMBL28221516 0.83 LMNA (0.58) LMNASMN1; SMN2HTTL3MBTL1MAPT
SCHEMBL527104 0.82 CTSK (0.64) CTSKKYNUCTSLCTSBCTSS
SCHEMBL527103 0.82 CTSK (0.64) CTSKKYNUCTSLCTSBCTSS
SCHEMBL4387860 0.82 CTSK (0.64) CTSKKYNUCTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113549074-A Triazole group-containing fused ring derivative inhibitor, and preparation method and application thereof 上海翰森生物医药科技有限公司 2021-10-26 CN disclosed
CN-113527307-A Triazole group-containing fused ring derivative inhibitor, and preparation method and application thereof 上海翰森生物医药科技有限公司 2021-10-22 CN disclosed