SCHEMBL28650118

SCHEMBL28650118

CCOC(=O)c1c(NC(=O)c2ccccc2)sc2c1CCC(C)C2

nearest known ligand 0.72

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.72
THRB P10828 2/20 0.66
MAPT P10636 8/20 0.65
TLR2 O60603 1/20 0.65
KDM4E B2RXH2 4/20 0.64
TNF P01375 2/20 0.63
NOD1 Q9Y239 2/20 0.63
HSD17B10 Q99714 2/20 0.63
ALDH1A1 P00352 2/20 0.63
NPSR1 Q6W5P4 2/20 0.63
LMNA P02545 2/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
MEN1 O00255 1/20 0.61
HPGD P15428 1/20 0.61
KMT2A Q03164 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28663924 0.92 ALDH1A1 (0.68) TP53THRBMAPTTLR2KDM4E
SCHEMBL28648841 0.89 THRB (0.82) TP53THRBMAPTKDM4EHSD17B10
SCHEMBL3913991 0.86 MAPT (0.66) TP53MAPTTLR2KDM4EHSD17B10
SCHEMBL2182372 0.84 TP53 (0.80) TP53THRBMAPTKDM4ETNF
SCHEMBL3916162 0.84 MAPT (0.80) TP53MAPTTLR2KDM4EHSD17B10
SCHEMBL8290510 0.84 MAPT (0.77) TP53MAPTTLR2KDM4EHSD17B10
SCHEMBL5807115 0.83 MAPT (0.71) TP53THRBMAPTTLR2KDM4E
SCHEMBL21333081 0.82 THRB (0.59) TP53THRBMAPTKDM4EHSD17B10
SCHEMBL12470159 0.82 MAPT (0.76) TP53MAPTTLR2KDM4EHSD17B10
SCHEMBL3914272 0.82 MAPT (0.58) TP53THRBMAPTKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113501807-A Tetrahydrobenzothiophene compound, and preparation method and application of pharmaceutical composition 重庆科技学院 2021-10-15 CN disclosed