SCHEMBL28650685

SCHEMBL28650685

COc1ncc(Cc2c(Cl)cc(O)cc2Cl)cc1C(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 8/20 0.43
THRA P10827 7/20 0.43
RORC P51449 3/20 0.38
DHFR P00374 1/20 0.33
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 2/20 0.32
MAPK1 P28482 1/20 0.31
P2RX3 P56373 1/20 0.30
P2RX2 Q9UBL9 1/20 0.30
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
RECQL P46063 1/20 0.30
KMT2A Q03164 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30083001 1.00 THRB (0.43) THRBTHRARORCDHFRCYP3A4
SCHEMBL24449953 0.87 THRB (0.38) THRBTHRARORCDHFRP2RX3
SCHEMBL28649667 0.79 THRA (0.38) THRBTHRARORCCYP3A4CYP2D6
SCHEMBL30083018 0.79 THRA (0.38) THRBTHRARORCCYP3A4CYP2D6
SCHEMBL24450105 0.78 RORC (0.37) THRBTHRARORCMAPTL3MBTL1
SCHEMBL28669913 0.78 THRA (0.41) THRBTHRARORCALDH1A1
SCHEMBL28650050 0.75 RORC (0.37) THRBRORCDHFRP2RX3P2RX2
SCHEMBL28668263 0.75 RORC (0.35) RORCCYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL30083017 0.75 RORC (0.35) RORCCYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL29527123 0.75 THRB (0.41) THRBTHRADHFRP2RX3P2RX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113698388-B 6-oxo-1, 6-dihydropyridine derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed
CN-113698388-A 6-oxo-1, 6-dihydropyridine derivatives, preparation method and application thereof in medicines 江苏恒瑞医药股份有限公司 2021-11-26 CN disclosed