SCHEMBL30083017

SCHEMBL30083017

COc1ncc(C(O)c2c(Cl)cc(O)cc2Cl)cc1C(C)C

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.35
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 2/20 0.32
MAPK1 P28482 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
P2RX3 P56373 1/20 0.31
P2RX2 Q9UBL9 1/20 0.31
LMNA P02545 1/20 0.30
GABRA1 P14867 1/20 0.30
GABRB1 P18505 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28668263 1.00 RORC (0.35) RORCCYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL24450006 0.78 RORC (0.38) RORCCYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL16133709 0.76 GABRA1 (0.35) RORCP2RX3P2RX2GABRA1
SCHEMBL28650685 0.75 THRB (0.43) RORCCYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL30083001 0.75 THRB (0.43) RORCCYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL22959247 0.74 PIK3R1 (0.35) RORCP2RX3P2RX2GABRA1GABRB1
SCHEMBL29527128 0.74 PIK3R1 (0.35) RORCP2RX3P2RX2GABRA1GABRB1
SCHEMBL29526921 0.71 RORC (0.35) RORCCYP3A4LMNA
SCHEMBL11890406 0.71 TSHR (0.43) RORCMAPK1P2RX3P2RX2LMNA
SCHEMBL12089821 0.68 SMN1; SMN2 (0.39) RORCCYP3A4CYP2D6SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113698388-B 6-oxo-1, 6-dihydropyridine derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed