SCHEMBL28655366

SCHEMBL28655366

SCc1cccc(-c2ccccc2)c1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.47
ALDH1A1 P00352 4/20 0.46
MAPK1 P28482 2/20 0.46
FOLH1 Q04609 3/20 0.46
PDCD1 Q15116 3/20 0.46
CD274 Q9NZQ7 3/20 0.46
IDO1 P14902 2/20 0.40
KMT2A Q03164 1/20 0.40
DCLRE1A Q6PJP8 1/20 0.37
DCLRE1B Q9H816 1/20 0.37
HSD17B10 Q99714 2/20 0.37
HPGD P15428 1/20 0.37
BCL2L1 Q07817 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB2 P47870 1/20 0.37
CYP2A6 P11509 1/20 0.37
HTR7 P34969 1/20 0.35
PTGER1 P34995 1/20 0.35
PTGER4 P35408 1/20 0.35
PTGER3 P43115 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29424918 0.83 DPP4 (0.47) DPP4ALDH1A1MAPK1FOLH1PDCD1
SCHEMBL30625954 0.83 PDCD1 (0.60) DPP4ALDH1A1MAPK1FOLH1PDCD1
SCHEMBL3392132 0.83 DPP4 (0.47) DPP4ALDH1A1MAPK1FOLH1PDCD1
SCHEMBL10982314 0.83 PDCD1 (0.60) DPP4ALDH1A1MAPK1FOLH1PDCD1
SCHEMBL2209528 0.82 DPP4 (0.60) DPP4ALDH1A1MAPK1FOLH1PDCD1
SCHEMBL27907921 0.82 GABRA1 (0.61) DPP4ALDH1A1MAPK1FOLH1PDCD1
SCHEMBL429933 0.79 ALDH1A1 (0.62) DPP4ALDH1A1MAPK1PDCD1CD274
SCHEMBL6701461 0.79 DPP4 (0.47) DPP4ALDH1A1MAPK1FOLH1PDCD1
SCHEMBL27900782 0.79 FOLH1 (0.50) DPP4ALDH1A1MAPK1FOLH1PDCD1
SCHEMBL6701464 0.78 DPP4 (0.50) DPP4ALDH1A1MAPK1FOLH1PDCD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113582971-B Small molecule immunosuppressant, preparation method and application thereof 北京康辰药业股份有限公司 2023-10-20 CN disclosed
CN-113582971-A Small molecule immunosuppressant, preparation method and application thereof 北京康辰药业股份有限公司 2021-11-02 CN disclosed