SCHEMBL28655835

SCHEMBL28655835

O=C(Oc1ccncn1)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.40
BRAF P15056 1/20 0.40
MAPK14 Q16539 1/20 0.40
TNNI3K Q59H18 1/20 0.40
HSP90AA1 P07900 1/20 0.36
P2RX7 Q99572 1/20 0.36
PLOD2 O00469 1/20 0.35
PLOD3 O60568 1/20 0.35
PLOD1 Q02809 1/20 0.35
HSD17B10 Q99714 1/20 0.32
GRM4 Q14833 1/20 0.30
CYP19A1 P11511 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30606641 0.82 ELANE (0.43) HSP90AA1P2RX7
SCHEMBL3657194 0.77 HSP90AA1 (0.41) KDRBRAFMAPK14TNNI3KHSP90AA1
SCHEMBL3170356 0.76 KDM4E (0.40)
Trifluoroacetic Acid SCHEMBL30271810 0.76 SLC22A12 (0.42) KDRBRAFMAPK14TNNI3KP2RX7
SCHEMBL8390998 0.76 HSP90AA1 (0.45) KDRBRAFMAPK14TNNI3KHSP90AA1
SCHEMBL12470613 0.76 HSP90AA1 (0.40) KDRBRAFMAPK14TNNI3KHSP90AA1
SCHEMBL2788170 0.76 P2RX7 (0.43) KDRBRAFMAPK14TNNI3KHSP90AA1
SCHEMBL29080505 0.74 HSP90AA1 (0.39) KDRBRAFMAPK14TNNI3KHSP90AA1
SCHEMBL30575119 0.74 HSP90AA1 (0.39) KDRBRAFMAPK14TNNI3KHSP90AA1
SCHEMBL30664890 0.73 HSD17B10 (0.48) KDRBRAFMAPK14TNNI3KPLOD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112996794-A Fused heterocyclic compounds as RET kinase inhibitors 阿雷生物药品公司 2021-06-18 CN disclosed