SCHEMBL2865597

SCHEMBL2865597

c1ccc(CNCc2cccc3ccccc23)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MC5R P33032 2/20 0.70
MAPK1 P28482 1/20 0.70
KMT2A Q03164 4/20 0.62
MEN1 O00255 3/20 0.62
MC1R Q01726 1/20 0.58
CYP1A2 P05177 2/20 0.56
CYP2D6 P10635 2/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
HSD17B10 Q99714 1/20 0.56
PKM P14618 1/20 0.55
HPGD P15428 1/20 0.54
CA2 P00918 2/20 0.50
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA4 P22748 1/20 0.49
CA9 Q16790 1/20 0.49
ALOX15 P16050 1/20 0.49
HIF1A Q16665 1/20 0.49
MAPT P10636 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30482193 1.00 MC5R (0.70) MC5RMAPK1KMT2AMEN1MC1R
SCHEMBL6008064 0.90 MC5R (0.70) MC5RMAPK1KMT2AMEN1MC1R
SCHEMBL3242373 0.86 MC5R (0.67) MC5RMAPK1KMT2AMEN1MC1R
SCHEMBL21296202 0.86 MC5R (0.67) MC5RMAPK1KMT2AMEN1MC1R
SCHEMBL15131007 0.86 MAPK1 (0.67) MC5RMAPK1KMT2AMEN1MC1R
SCHEMBL15130991 0.86 MC5R (0.67) MC5RMAPK1KMT2AMEN1MC1R
SCHEMBL9080754 0.85 MC5R (0.66) MC5RMAPK1KMT2AMEN1MC1R
Hydrochloric Acid SCHEMBL31146828 0.84 MC5R (0.65) MC5RMAPK1KMT2AMEN1MC1R
SCHEMBL2343213 0.84 HPGD (0.62) MC5RMAPK1KMT2AMEN1HPGD
SCHEMBL15131004 0.84 CA12 (0.68) MC5RMAPK1KMT2AMEN1MC1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 58 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102834379-A Tricyclic indole derivatives as PBR ligands GE HEALTHCARE LTD 2012-12-19 CN claimed
US-20020107406-A1 Calcium receptor-active compounds NPS PHARMACEUTICALS, INC. (US) 2002-08-08 US claimed
EP-0933354-A1 CALCIUM RECEPTOR-ACTIVE COMPOUNDS KIRIN BEER KABUSHIKI KAISHA (JP) 1999-08-04 EP claimed
US-20250136594-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. 2025-05-01 US disclosed
EP-4469438-A1 COMPOUNDS AND METHODS OF USE Tango Therapeutics, Inc. (US) 2024-12-04 EP disclosed
US-12083140-B2 Pharmaceutical composition for preventing and treating glaucoma, containing adenosine derivative FUTURE MEDICINE CO., LTD. (KR) 2024-09-10 US disclosed
EP-3603647-B1 PHARMACEUTICAL COMPOSITION FOR PREVENTING AND TREATING GLAUCOMA, CONTAINING ADENOSINE DERIVATIVE FUTURE MEDICINE CO LTD (KR) 2024-08-21 EP disclosed
WO-2023146987-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. (US) 2023-08-03 WO disclosed
WO-2023146987-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. (US) 2023-08-03 WO disclosed
US-20210386771-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING AND TREATING GLAUCOMA, CONTAINING ADENOSINE DERIVATIVE FUTURE MEDICINE CO., LTD. (KR) 2021-12-16 US disclosed
US-11185556-B2 Pharmaceutical composition for preventing and treating glaucoma, containing adenosine derivative FUTURE MEDICINE CO., LTD. (KR) 2021-11-30 US disclosed
EP-0585202-A1 N,N'-alkenylene amine/mercaptotolyl-imidazole blends as high temperature antioxidants for elastomers CIBA-GEIGY AG (CH) 1994-03-02 EP disclosed
US-5283367-A Antioxidants for lubricants and polymers CIBA-GEIGY CORPORATION (US) 1994-02-01 US disclosed
US-5240976-A For automobile, wire and cable uses CIBA-GEIGY CORPORATION (US) 1993-08-31 US disclosed
US-5196164-A During addition polymerization, wall coating of anionic dye and cationic dye and organonitrogen compound SHIN-ETSU CHEMICAL CO., LTD. (JP) 1993-03-23 US disclosed
EP-0514333-A2 Substituted 1,4-diamino-2-butene stabilizers and stabilized compositions CIBA-GEIGY AG (CH) 1992-11-19 EP disclosed
EP-0355575-A2 Method of preventing polymer scale formation Shin-Etsu Chemical Co., Ltd. (JP) 1990-02-28 EP disclosed
US-4758639-A Process for production of vinyl polymer SHIN-ETSU CHEMICAL CO., LTD. (JP) 1988-07-19 US disclosed
US-4757124-A Suspension or emulsion polymerizing vinyl chloride monomer or mixture of vinyl chloride with vinyl monomer copolymerizable therewith in reactor with walls coated with antiscaling compound containing dye or pigments SHIN-ETSU CHEMICAL CO., LTD. (JP) 1988-07-12 US disclosed
EP-0172427-A2 Process for production of vinyl chloride polymer Shin-Etsu Chemical Co., Ltd. (JP) 1986-02-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250136594-A1 COMPOUNDS AND METHODS OF USE CNKSR1, UGT1A1, REV1 MC5R 553/4885MAPK1 3230/4885KMT2A 2276/4885
US-11185556-B2 Pharmaceutical composition for preventing and treating glaucoma, containing adenosine derivative ADORA1, ADORA2A, PDE3A MC5R 993/4885MAPK1 651/4885KMT2A 4100/4885
US-12083140-B2 Pharmaceutical composition for preventing and treating glaucoma, containing adenosine derivative ADORA1, ADORA2A, ADORA3 MC5R 1034/4885MAPK1 721/4885KMT2A 4047/4885
US-20210386771-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING AND TREATING GLAUCOMA, CONTAINING ADENOSINE DERIVATIVE ADORA1, ADORA2A, ADORA3 MC5R 1034/4885MAPK1 721/4885KMT2A 4047/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.