SCHEMBL28658071

SCHEMBL28658071

Brc1ccc(-c2[c]c(-c3ccccc3)sn2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
MAPK1 P28482 2/20 0.47
NR1H4 Q96RI1 1/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
NR1H2 P55055 3/20 0.36
NR1H3 Q13133 3/20 0.36
DGAT1 O75907 1/20 0.36
MAPK13 O15264 2/20 0.35
GCGR P47871 2/20 0.35
MAPK12 P53778 2/20 0.35
MAPK11 Q15759 2/20 0.35
MAPK14 Q16539 2/20 0.35
AGTR1 P30556 1/20 0.35
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28476983 0.89 ADORA3 (0.35) ALDH1A1MAPK1NPC1RAB9ASMN1; SMN2
SCHEMBL28655309 0.83 NPC1 (0.42) ALDH1A1NPC1RAB9ASMN1; SMN2NFKB1
SCHEMBL28653098 0.83 CYP1A2 (0.47) ALDH1A1NPC1RAB9ASMN1; SMN2NFKB1
SCHEMBL28650363 0.83 ALOX5 (0.37) ALDH1A1MAPK1NPC1RAB9ASMN1; SMN2
SCHEMBL435137 0.83 CYP1A2 (0.47) ALDH1A1NPC1RAB9ASMN1; SMN2NFKB1
SCHEMBL28661674 0.83 NPC1 (0.42) ALDH1A1NPC1RAB9ASMN1; SMN2NFKB1
SCHEMBL28650268 0.83 ALOX5 (0.37) ALDH1A1MAPK1NPC1RAB9ASMN1; SMN2
SCHEMBL28650037 0.79 TP53 (0.39) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL28661681 0.79 KIF11 (0.52) ALDH1A1DGAT1MAPK13MAPK12MAPK11
SCHEMBL28647365 0.79 KIF11 (0.52) ALDH1A1DGAT1MAPK13MAPK12MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111233783-B Synthetic method of isothiazol-4-yl disulfide derivative 温州大学 2021-11-16 CN disclosed
CN-111233783-A Synthesis method of bithiazole-4-yl disulfide derivative 温州大学 2020-06-05 CN disclosed