SCHEMBL435137

SCHEMBL435137

Clc1ccc(-c2[c]c(-c3ccccc3)sn2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
LMNA P02545 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
NPSR1 Q6W5P4 2/20 0.37
ALDH1A1 P00352 2/20 0.37
USP2 O75604 1/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
ADORA3 P0DMS8 2/20 0.36
NR1H2 P55055 2/20 0.36
NR1H3 Q13133 2/20 0.36
SCN2A Q99250 1/20 0.36
HTT P42858 1/20 0.36
ADORA2A P29274 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28653098 1.00 CYP1A2 (0.47) CYP1A2NPC1RAB9ALMNAL3MBTL1
SCHEMBL28476983 0.89 ADORA3 (0.35) NPC1RAB9AL3MBTL1ALDH1A1ADORA3
SCHEMBL28655312 0.83 NPC1 (0.42) NPC1RAB9ATSHRSCN2AADORA2A
SCHEMBL28655309 0.83 NPC1 (0.42) NPC1RAB9ALMNAL3MBTL1KDM4E
SCHEMBL28650363 0.83 ALOX5 (0.37) NPC1RAB9ALMNAL3MBTL1KDM4E
SCHEMBL28650268 0.83 ALOX5 (0.37) NPC1RAB9ALMNAL3MBTL1KDM4E
SCHEMBL28661674 0.83 NPC1 (0.42) NPC1RAB9ALMNAL3MBTL1KDM4E
SCHEMBL28658071 0.83 ALDH1A1 (0.47) NPC1RAB9ALMNAL3MBTL1KDM4E
SCHEMBL28586105 0.79 NPC1 (0.47) NPC1RAB9ALMNAL3MBTL1KDM4E
SCHEMBL28647365 0.79 KIF11 (0.52) ALDH1A1TSHRSCN2AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111233783-B Synthetic method of isothiazol-4-yl disulfide derivative 温州大学 2021-11-16 CN disclosed
CN-111233783-A Synthesis method of bithiazole-4-yl disulfide derivative 温州大学 2020-06-05 CN disclosed
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed