SCHEMBL28661992

SCHEMBL28661992

Cc1ccc(-c2noc(-c3ccc(F)c(O)c3)n2)cn1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.52
CHRNA5 P30532 1/20 0.52
CHRNA4 P43681 1/20 0.52
S1PR1 P21453 4/20 0.48
ADORA3 P0DMS8 1/20 0.48
ACHE P22303 4/20 0.45
PTGS2 P35354 1/20 0.43
TP53 P04637 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31657612 0.88 CHRNB2 (0.67) CHRNB2CHRNA5CHRNA4S1PR1ADORA3
SCHEMBL28653849 0.86 S1PR1 (0.63) S1PR1ADORA3TP53SMN1; SMN2ALDH1A1
SCHEMBL28659795 0.86 S1PR1 (0.50) CHRNB2CHRNA5CHRNA4S1PR1ADORA3
SCHEMBL28665259 0.84 ADORA3 (0.54) S1PR1ADORA3ACHETP53SMN1; SMN2
SCHEMBL28656184 0.84 S1PR1 (0.48) CHRNB2CHRNA5CHRNA4S1PR1ADORA3
SCHEMBL28654921 0.82 NPC1 (0.56) S1PR1SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL1423251 0.82 CHRNB2 (0.78) CHRNB2CHRNA5CHRNA4S1PR1TP53
SCHEMBL28664805 0.80 ADORA3 (0.52) CHRNB2CHRNA5CHRNA4S1PR1ADORA3
SCHEMBL28661994 0.78 GRM5 (0.45) CHRNB2CHRNA5CHRNA4S1PR1TP53
SCHEMBL30688269 0.77 MAPT (0.45) CHRNB2CHRNA5CHRNA4S1PR1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113603684-B 1,2, 4-oxadiazole Nrf2 activator-tac Lin Pinge product and preparation method and application thereof 中国药科大学 2023-12-19 CN disclosed
CN-113603684-A 1,2, 4-oxadiazole Nrf2 activator-tacrine split product and preparation method and application thereof 中国药科大学 2021-11-05 CN disclosed