SCHEMBL28664805

SCHEMBL28664805

Cc1ccc(-c2noc(-c3cccc(O)c3)n2)cn1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.52
TP53 P04637 2/20 0.50
ALDH1A1 P00352 1/20 0.50
NFKB1 P19838 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
ACHE P22303 1/20 0.48
S1PR1 P21453 2/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
HAVCR2 Q8TDQ0 1/20 0.48
MAPT P10636 3/20 0.47
CHRNB2 P17787 2/20 0.47
CHRNA5 P30532 2/20 0.47
CHRNA4 P43681 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28653849 0.82 S1PR1 (0.63) ADORA3TP53ALDH1A1NFKB1NFKB2
SCHEMBL28659795 0.82 S1PR1 (0.50) ADORA3TP53ALDH1A1NFKB1NFKB2
SCHEMBL8039918 0.82 CHRNB2 (0.71) TP53ALDH1A1NFKB1NFKB2RELA
SCHEMBL12643444 0.81 NR1H4 (0.53) TP53ALDH1A1NFKB1NFKB2RELA
SCHEMBL1422802 0.81 CHRNB2 (0.71) ADORA3TP53ALDH1A1NFKB1NFKB2
SCHEMBL28661992 0.80 CHRNB2 (0.52) ADORA3TP53ALDH1A1NFKB1NFKB2
SCHEMBL28656184 0.80 S1PR1 (0.48) ADORA3TP53ALDH1A1NFKB1NFKB2
SCHEMBL28665259 0.80 ADORA3 (0.54) ADORA3TP53ALDH1A1NFKB1NFKB2
SCHEMBL7958582 0.79 NR1H4 (0.67) TP53ALDH1A1NFKB1NFKB2RELA
SCHEMBL21228152 0.79 HSD17B2 (0.66)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113603684-B 1,2, 4-oxadiazole Nrf2 activator-tac Lin Pinge product and preparation method and application thereof 中国药科大学 2023-12-19 CN disclosed
CN-113603684-A 1,2, 4-oxadiazole Nrf2 activator-tacrine split product and preparation method and application thereof 中国药科大学 2021-11-05 CN disclosed