SCHEMBL28665259

SCHEMBL28665259

Cc1ccc(-c2noc(-c3ccc(Cl)c(O)c3)n2)cn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.54
S1PR1 P21453 3/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA9 Q16790 1/20 0.48
NPC1 O15118 4/20 0.47
RAB9A P51151 4/20 0.47
ACHE P22303 2/20 0.45
NR1H4 Q96RI1 1/20 0.43
TP53 P04637 4/20 0.43
MAPT P10636 4/20 0.43
MEN1 O00255 1/20 0.43
PKM P14618 1/20 0.43
TSHR P16473 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
MAPK1 P28482 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28653849 0.86 S1PR1 (0.63) ADORA3S1PR1NPC1RAB9ATP53
SCHEMBL28659795 0.86 S1PR1 (0.50) ADORA3S1PR1NPC1RAB9AACHE
SCHEMBL28661992 0.84 CHRNB2 (0.52) ADORA3S1PR1NPC1RAB9AACHE
SCHEMBL28656184 0.84 S1PR1 (0.48) ADORA3S1PR1NPC1RAB9AACHE
SCHEMBL28654921 0.82 NPC1 (0.56) S1PR1NPC1RAB9AMAPTTSHR
SCHEMBL28664805 0.80 ADORA3 (0.52) ADORA3S1PR1NPC1RAB9AACHE
SCHEMBL28665260 0.78 NPC1 (0.51) S1PR1CA12CA1CA2CA9
SCHEMBL31657612 0.77 CHRNB2 (0.67) ADORA3S1PR1NPC1RAB9AACHE
SCHEMBL30688270 0.77 ADORA3 (0.49) ADORA3S1PR1NPC1RAB9AACHE
SCHEMBL28659723 0.77 ADORA3 (0.49) ADORA3S1PR1NPC1RAB9AACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113603684-B 1,2, 4-oxadiazole Nrf2 activator-tac Lin Pinge product and preparation method and application thereof 中国药科大学 2023-12-19 CN disclosed
CN-113603684-A 1,2, 4-oxadiazole Nrf2 activator-tacrine split product and preparation method and application thereof 中国药科大学 2021-11-05 CN disclosed