SCHEMBL286704

SCHEMBL286704

Cc1cc(Cl)ncc1C#N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 1/20 0.46
CSNK1A1 P48729 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
ALDH1A1 P00352 4/20 0.40
IDH1 O75874 2/20 0.37
S1PR1 P21453 1/20 0.37
S1PR3 Q99500 1/20 0.37
NPSR1 Q6W5P4 3/20 0.37
TDP1 Q9NUW8 1/20 0.37
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.35
SRC P12931 2/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
LRRK2 Q5S007 1/20 0.35
EGFR P00533 1/20 0.35
ERBB2 P04626 1/20 0.35
CYP11B2 P19099 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31750396 1.00 S1PR2 (0.46) S1PR2CSNK1A1CLK4ALDH1A1IDH1
SCHEMBL19565835 0.83 ALDH1A1 (0.40) S1PR2CSNK1A1CLK4ALDH1A1S1PR1
SCHEMBL29505699 0.78 UHRF1 (0.46) S1PR2CSNK1A1CLK4ALDH1A1IDH1
SCHEMBL317517 0.78 UHRF1 (0.46) S1PR2CSNK1A1CLK4ALDH1A1IDH1
SCHEMBL30445578 0.78 CSNK1A1 (0.44) CSNK1A1CLK4ALDH1A1NPSR1TDP1
SCHEMBL1286023 0.78 CSNK1A1 (0.44) CSNK1A1CLK4ALDH1A1NPSR1TDP1
SCHEMBL21927619 0.77 EGLN2 (0.41) S1PR2CSNK1A1CLK4ALDH1A1IDH1
SCHEMBL5555501 0.76 GPBAR1 (0.45) ALDH1A1NPSR1TDP1TSHRLRRK2
SCHEMBL14068317 0.75 S1PR2 (0.37) S1PR2CSNK1A1CLK4ALDH1A1IDH1
SCHEMBL21296119 0.75 CSNK1A1 (0.41) S1PR2CSNK1A1CLK4ALDH1A1S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 85 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12570671-B2 Substituted oxoisoindoline compounds for the treatment of cancer BRISTOL-MYERS SQUIBB COMPANY (US) 2026-03-10 US disclosed
US-20260055094-A1 FXR (NR1H4) MODULATING COMPOUNDS GILEAD SCIENCES INC (US) 2026-02-26 US disclosed
EP-4126843-B1 SUBSTITUTED OXOISOINDOLINE COMPOUNDS FOR THE TREATMENT OF CANCER BRISTOL MYERS SQUIBB CO (US) 2026-02-11 EP disclosed
US-12358903-B2 FXR (NR1H4) modulating compounds GILEAD SCIENCES, INC. (US) 2025-07-15 US disclosed
US-20240383853-A1 OXIMES AND THEIR USE IN TREATMENT OF GBA-RELATED DISEASES Zevra Denmark A/S (DK) 2024-11-21 US disclosed
CN-115605466-B Substituted oxoisoindoline compounds for the treatment of cancer 百时美施贵宝公司 2024-11-01 CN disclosed
EP-4408533-A1 OXIMES AND THEIR USE IN TREATMENT OF GBA-RELATED DISEASES Zevra Denmark A/S (DK) 2024-08-07 EP disclosed
CN-118139842-A Oximes and their use in the treatment of GBA related diseases 泽拉丹麦有限公司 2024-06-04 CN disclosed
WO-2024003773-A1 2,7-NAPHTHYRIDINE COMPOUNDS AS MASTL INHIBITORS PFIZER INC. (US) 2024-01-04 WO disclosed
US-20230322803-A1 SUBSTITUTED OXOISOINDOLINE COMPOUNDS FOR THE TREATMENT OF CANCER BRISTOL MYERS SQUIBB CO (US) 2023-10-12 US disclosed
US-20140142115-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2014-05-22 US disclosed
US-8673920-B2 Inhibitors of the renal outer medullary potassium channel MERCK SHARP & DOHME CORP. (US) 2014-03-18 US disclosed
EP-2427444-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL Merck Sharp & Dohme Corp. (US) 2012-03-14 EP disclosed
WO-2010129379-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2010-11-11 WO disclosed
US-20100286123-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME LLC 2010-11-11 US disclosed
EP-1999110-B1 PROCESS FOR PREPARING l-HALO-2,7-NAPHTHYRIDINYL DERIVATIVES UCB PHARMA SA (BE) 2009-09-16 EP disclosed
US-20090221828-A1 Process for Preparing 1-Halo-2,7-Naphthyridinyl Derivatives UCB PHARMA, S.A. (BE) 2009-09-03 US disclosed
US-7528140-B2 Substituted pyrrolo[3,2-d]pyrimidines as glycogen synthase kinase (GSK) inhibitors TEIJIN LIMITED (JP) 2009-05-05 US disclosed
EP-1999110-A2 PROCESS FOR PREPARING l-HALO-2,7-NAPHTHYRIDINYL DERIVATIVES UCB Pharma, S.A. (BE) 2008-12-10 EP disclosed
WO-2007107345-A2 PROCESS FOR PREPARING l-HALO-2,7-NAPHTHYRIDINYL DERIVATIVES UCB PHARMA, S.A. (BE) 2007-09-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12358903-B2 FXR (NR1H4) modulating compounds NR1H4, NR1H2, NR1H3 S1PR2 410/4885CSNK1A1 2680/4885CLK4 3976/4885
US-20230322803-A1 SUBSTITUTED OXOISOINDOLINE COMPOUNDS FOR THE TREATMENT OF CANCER DDX21, HRAS, RPL17 S1PR2 2945/4885CSNK1A1 963/4885CLK4 4846/4885
US-12570671-B2 Substituted oxoisoindoline compounds for the treatment of cancer NR3C1, NR2C2, RIOX2 S1PR2 760/4885CSNK1A1 833/4885CLK4 4805/4885
US-20240383853-A1 OXIMES AND THEIR USE IN TREATMENT OF GBA-RELATED DISEASES GBA1, GBA2, GBA3 S1PR2 741/4885CSNK1A1 3479/4885CLK4 4388/4885
US-20140142115-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL KCNJ11, KCNJ1, KCNJ2 S1PR2 1180/4885CSNK1A1 1572/4885CLK4 869/4885
US-20260055094-A1 FXR (NR1H4) MODULATING COMPOUNDS NR1H4, NR1H2, NR1H3 S1PR2 450/4885CSNK1A1 709/4885CLK4 3530/4885
US-20090221828-A1 Process for Preparing 1-Halo-2,7-Naphthyridinyl Derivatives NPM1, XPO4, BRD7 S1PR2 4518/4885CSNK1A1 395/4885CLK4 281/4885
US-20100286123-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL KCNJ11, KCNJ1, KCNJ2 S1PR2 1180/4885CSNK1A1 1572/4885CLK4 869/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.