SCHEMBL28682189

SCHEMBL28682189

N=c1ccc2cccc(Br)c2[nH]1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.60
CA9 Q16790 3/20 0.60
NOS1 P29475 1/20 0.42
HRH4 Q9H3N8 1/20 0.35
BACE1 P56817 1/20 0.34
KDM4E B2RXH2 1/20 0.33
HSD17B10 Q99714 1/20 0.33
AR P10275 1/20 0.33
NISCH Q9Y2I1 1/20 0.31
ENPP3 O14638 1/20 0.31
ENPP1 P22413 1/20 0.31
DYRK1A Q13627 3/20 0.31
CDK9 P50750 1/20 0.30
DYRK2 Q92630 1/20 0.30
DYRK1B Q9Y463 1/20 0.30
CLK1 P49759 1/20 0.30
GSK3B P49841 1/20 0.30
CDK5 Q00535 1/20 0.30
CDK5R1 Q15078 1/20 0.30
MEN1 O00255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL731556 0.75 CA12 (1.00) CA12CA9NOS1HRH4BACE1
SCHEMBL21877855 0.70 CA12 (0.53) CA12CA9NOS1HRH4BACE1
SCHEMBL17673224 0.68 CA12 (0.52) CA12CA9NOS1HRH4BACE1
SCHEMBL341141 0.67 ALDH1A1 (0.49) KDM4EHSD17B10ARMEN1GAA
SCHEMBL445281 0.67 AHR (0.56) CA12CA9NOS1BACE1AR
SCHEMBL597517 0.67 CA12 (0.50) CA12CA9NOS1HRH4KDM4E
SCHEMBL6505957 0.67 CA12 (0.50) CA12CA9NOS1HRH4BACE1
SCHEMBL17722736 0.64 KIF11 (0.58) CA12CA9NOS1KDM4EHSD17B10
SCHEMBL29597557 0.64 ALDH1A1 (0.54) CA12CA9KDM4EHSD17B10MEN1
SCHEMBL403269 0.64 ALDH1A1 (0.54) CA12CA9KDM4EHSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114989137-B Chiral imine-containing quinoline imidazoline compound and metal complex thereof, preparation method and application 浙江大学 2024-03-01 CN disclosed
CN-113880822-B Chiral imine quinoline oxazoline-containing compound and metal complex thereof, preparation method and application 浙江大学 2023-09-19 CN disclosed
CN-113880822-A Chiral quinoline oxazoline compound containing imine and metal complex thereof, and preparation method and application thereof 浙江大学 2022-01-04 CN disclosed