SCHEMBL28690109

SCHEMBL28690109

COc1ccc(C(=O)C=[N+]=[N-])cn1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NNMT P40261 2/20 0.57
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
ALDH1A1 P00352 3/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
HTT P42858 2/20 0.49
HIF1A Q16665 1/20 0.49
MKNK1 Q9BUB5 1/20 0.48
MKNK2 Q9HBH9 1/20 0.48
GPR183 P32249 5/20 0.41
MAPT P10636 2/20 0.41
OXTR P30559 1/20 0.40
KCNH2 Q12809 1/20 0.39
KDM4E B2RXH2 2/20 0.39
SIRT6 Q8N6T7 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30474575 1.00 NNMT (0.57) NNMTMAOAMAOBALDH1A1MEN1
SCHEMBL9672055 0.79 ALDH1A1 (0.49) NNMTALDH1A1MEN1KMT2AHTT
SCHEMBL10123137 0.79 KMT2A (0.53) ALDH1A1MEN1KMT2AHTTHIF1A
SCHEMBL4582774 0.76 NNMT (0.58) NNMTMAOAMAOBALDH1A1MEN1
SCHEMBL4582780 0.76 NNMT (0.58) NNMTMAOAMAOBALDH1A1MEN1
SCHEMBL18228074 0.76 NNMT (0.72) NNMTMAOAMAOBALDH1A1MEN1
SCHEMBL27313612 0.75 NNMT (0.66) NNMTMAOAMAOBALDH1A1HTT
SCHEMBL9449259 0.75 ALDH1A1 (0.61) MAOAMAOBALDH1A1MEN1KMT2A
SCHEMBL29757598 0.74 NNMT (0.70) NNMTALDH1A1MKNK1MKNK2MAPT
SCHEMBL29514668 0.74 NNMT (0.70) NNMTMAOAMAOBALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354635-B Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2023-04-18 CN disclosed
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed