SCHEMBL9449259

SCHEMBL9449259

COc1ccc(C(=O)C=[N+]=[N-])cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.61
MEN1 O00255 3/20 0.61
KMT2A Q03164 3/20 0.61
HTT P42858 1/20 0.61
HIF1A Q16665 1/20 0.61
F3 P13726 2/20 0.54
CES2 O00748 1/20 0.53
CES1 P23141 1/20 0.53
MAPT P10636 5/20 0.53
HPGD P15428 1/20 0.53
CA1 P00915 4/20 0.52
CA2 P00918 4/20 0.52
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C19 P33261 1/20 0.51
MAOB P27338 4/20 0.50
HSPD1 P10809 1/20 0.50
TNFRSF1A P19438 1/20 0.50
HSPE1 P61604 1/20 0.50
CYP1B1 Q16678 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20134914 0.81 ALDH1A1 (0.61) ALDH1A1MEN1KMT2AHTTHIF1A
SCHEMBL9449106 0.81 ABCG2 (0.53) ALDH1A1MEN1KMT2AHTTHIF1A
SCHEMBL9448934 0.81 KMT2A (0.56) ALDH1A1MEN1KMT2AHTTHIF1A
SCHEMBL9448898 0.80 ABCG2 (0.59) ALDH1A1MEN1KMT2AHTTCES2
SCHEMBL9448941 0.79 ALDH1A1 (0.54) ALDH1A1MEN1KMT2AHTTHIF1A
SCHEMBL9449020 0.79 ALDH1A1 (0.67) ALDH1A1MEN1KMT2AHTTHIF1A
SCHEMBL7000261 0.78 F3 (0.75) ALDH1A1MEN1KMT2AF3CES2
SCHEMBL7000262 0.78 F3 (0.75) ALDH1A1MEN1KMT2AF3CES2
SCHEMBL4607255 0.77 KMT2A (0.56) ALDH1A1MEN1KMT2AHTTHIF1A
SCHEMBL28111426 0.76 CES2 (0.61) ALDH1A1MEN1KMT2AF3CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248458-B Preparation method of alpha-carbonyl amide compound 陕西省煤田地质集团有限公司 2022-09-27 CN disclosed
CN-113248458-A Preparation method of alpha-carbonyl amide compound 陕西省煤田地质集团有限公司 2021-08-13 CN disclosed
US-9751825-B2 TAK1 kinase inhibitors, compositions, and used related thereto EMORY UNIVERSITY (US) 2017-09-05 US disclosed
US-20140249199-A1 TAK1 KINASE INHIBITORS, COMPOSITIONS, AND USED RELATED THERETO HEALTH RESEARCH, INC. (US) 2014-09-04 US disclosed
EP-0466730-B1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1993-07-21 EP disclosed
US-5220021-A Geminal bisphosphonic acids and derivatives as anti-arthritic agents THE UPJOHN COMPANY (US) 1993-06-15 US disclosed
WO-1990012017-A1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1990-10-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140249199-A1 TAK1 KINASE INHIBITORS, COMPOSITIONS, AND USED RELATED THERETO TAB1, MAP3K1, MAP3K6 ALDH1A1 3574/4885MEN1 1525/4885KMT2A 1834/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.