SCHEMBL28690110

SCHEMBL28690110

NC(=O)Oc1cc2ccc(Br)cc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.42
AHR P35869 2/20 0.41
CYP2A6 P11509 1/20 0.37
NR4A2 P43354 1/20 0.37
NCEH1 Q6PIU2 1/20 0.36
GPR183 P32249 2/20 0.36
NOS1 P29475 1/20 0.35
METAP2 P50579 1/20 0.35
DYRK1A Q13627 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29056767 0.87 FLT3 (0.47) HRH4AHRCYP2A6NR4A2NCEH1
SCHEMBL3381701 0.85 HRH4 (0.43) HRH4AHRNCEH1
SCHEMBL3836490 0.78 FLT3 (0.50) CYP2A6
SCHEMBL8889640 0.75 HRH4 (0.55) HRH4GPR183
SCHEMBL4036292 0.73 DAO (0.50) HRH4DYRK1A
SCHEMBL3381954 0.72 FLT3 (0.48) HRH4AHRCYP2A6NR4A2NCEH1
SCHEMBL25305363 0.70 NCEH1 (0.62) CYP2A6NCEH1
SCHEMBL13504611 0.70 PDPK1 (0.40) METAP2DYRK1A
SCHEMBL4033217 0.70 DAO (0.50) HRH4DYRK1A
SCHEMBL19611005 0.70 DRD4 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115943144-A Compound serving as PAK4 kinase inhibitor and preparation method and application thereof 成都海博为药业有限公司 2023-04-07 CN disclosed
CN-114075175-A Compound serving as PAK4 kinase inhibitor and preparation method and application thereof 成都海博为药业有限公司 2022-02-22 CN disclosed