SCHEMBL28690666

SCHEMBL28690666

Cc1ccccc1CC(=O)Nc1ccc(=O)n(-c2ccccc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.52
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
NPC1 O15118 2/20 0.47
AKR1B1 P15121 1/20 0.46
CYP1A2 P05177 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
BLM P54132 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CACNA1G O43497 1/20 0.45
CACNA1H O95180 1/20 0.45
CACNA1I Q9P0X4 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
P2RY14 Q15391 1/20 0.43
MAPK8 P45983 1/20 0.43
ANO1 Q5XXA6 1/20 0.42
ROCK2 O75116 1/20 0.42
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28706311 0.88 ALDH1A1 (0.48) TDP1KMT2AMEN1NPC1CYP1A2
SCHEMBL28708127 0.88 CA12 (0.53) KMT2AMEN1CYP1A2KDM4EALDH1A1
SCHEMBL28697076 0.85 ELOVL1 (0.52) KMT2AMEN1NPC1CYP1A2ALDH1A1
SCHEMBL28684562 0.85 KCNJ5 (0.56) NPC1KDM4EALDH1A1MAPK8LMNA
SCHEMBL28704823 0.84 MEN1 (0.57) KMT2AMEN1KDM4EALDH1A1HPGD
SCHEMBL28706294 0.83 KMT2A (0.58) KMT2AMEN1KDM4EALDH1A1HPGD
SCHEMBL28697085 0.83 KDM4E (0.47) KMT2AMEN1NPC1CYP1A2KDM4E
SCHEMBL28698365 0.82 ALDH1A1 (0.52) KMT2AMEN1CYP1A2KDM4EALDH1A1
SCHEMBL28690641 0.82 NR2E1 (0.51) KMT2AMEN1CYP1A2ANO1CYP2D6
SCHEMBL28933313 0.80 MEN1 (0.54) KMT2AMEN1CYP1A2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114057630-B Pirfenidone derivative and synthetic method and application thereof 郑州大学 2023-06-02 CN claimed
CN-114057630-A Pirfenidone derivative and synthetic method and application thereof 郑州大学 2022-02-18 CN claimed
CN-114057630-B Pirfenidone derivative and synthetic method and application thereof 郑州大学 2023-06-02 CN disclosed
CN-114057630-A Pirfenidone derivative and synthetic method and application thereof 郑州大学 2022-02-18 CN disclosed