SCHEMBL2869092

SCHEMBL2869092

COc1ccc(CCNS(=O)(=O)c2cc(-c3[nH]c4ccccc4c3C(=O)C(=O)O)ccc2Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
ALOX5 P09917 1/20 0.49
POLB P06746 3/20 0.49
SMN1; SMN2 Q16637 1/20 0.45
AKR1C3 P42330 1/20 0.44
MAPT P10636 3/20 0.44
LMNA P02545 1/20 0.44
CNR1 P21554 1/20 0.43
SGMS1 Q86VZ5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2873354 0.93 ALDH1A1 (0.52) ALDH1A1ALOX5POLBSMN1; SMN2AKR1C3
SCHEMBL3998593 0.88 ALDH1A1 (0.50) ALDH1A1ALOX5POLBSMN1; SMN2AKR1C3
SCHEMBL2875353 0.88 ALOX5 (0.55) ALDH1A1ALOX5POLBSMN1; SMN2AKR1C3
SCHEMBL2878276 0.88 MAPT (0.48) ALDH1A1ALOX5POLBSMN1; SMN2MAPT
SCHEMBL2878351 0.86 ALOX5 (0.55) ALDH1A1ALOX5MAPT
SCHEMBL2873169 0.85 ACLY (0.51) ALDH1A1ALOX5POLBSMN1; SMN2AKR1C3
SCHEMBL2873564 0.83 MAPT (0.44) ALDH1A1ALOX5POLBMAPT
SCHEMBL2878384 0.81 MAPT (0.48) ALDH1A1ALOX5MAPT
SCHEMBL3998451 0.80 ACLY (0.50) ALDH1A1ALOX5SMN1; SMN2AKR1C3MAPT
SCHEMBL2872278 0.80 ACLY (0.51) ALDH1A1ALOX5SMN1; SMN2AKR1C3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2066628-B1 2-PHENYL-INDOLES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2010-10-20 EP disclosed