SCHEMBL286951

SCHEMBL286951

COCCOC(=O)C1=CN=CC(CC(=O)c2ccc(Cl)cc2Cl)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
MAPK1 P28482 2/20 0.37
HIF1A Q16665 1/20 0.37
KMT2A Q03164 3/20 0.37
AGTR1 P30556 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MEN1 O00255 1/20 0.37
HTT P42858 1/20 0.37
KDM4E B2RXH2 2/20 0.35
RECQL P46063 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPC1 O15118 1/20 0.35
TSHR P16473 1/20 0.34
ERCC5 P28715 1/20 0.34
FEN1 P39748 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL286991 0.84 SMN1; SMN2 (0.40) ALDH1A1MAPK1HIF1AKMT2AAGTR1
SCHEMBL287785 0.80 SMN1; SMN2 (0.41) ALDH1A1MAPK1HIF1AKMT2AAGTR1
SCHEMBL287667 0.74 ALDH1A1 (0.32) ALDH1A1MAPK1HIF1AKMT2AL3MBTL1
SCHEMBL287282 0.71 TDP1 (0.43) ALDH1A1MAPK1HIF1AKMT2AL3MBTL1
SCHEMBL660547 0.70 ALDH1A1 (0.39) ALDH1A1MAPK1HIF1AKMT2AAGTR1
SCHEMBL287683 0.66 NPC1 (0.39) ALDH1A1KMT2AMEN1KDM4ECYP1A2
SCHEMBL31114507 0.64 ALDH1A1 (0.62) ALDH1A1MAPK1HIF1AKMT2AAGTR1
SCHEMBL6227326 0.64 GLA (0.48) ALDH1A1MAPK1HIF1AKMT2AAGTR1
Bromide SCHEMBL1194556 0.63 GLA (0.50) ALDH1A1MAPK1HIF1AKMT2AAGTR1
SCHEMBL6941866 0.63 TSHR (0.53) ALDH1A1MAPK1KMT2AKDM4ERECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427432-A2 NOVEL HETEROCYCLIC COMPOUNDS Torrent Pharmaceuticals Limited (IN) 2012-03-14 EP claimed
WO-2010128528-A2 NOVEL HETEROCYCLIC COMPOUNDS TORRENT PHARMACEUTICALS LIMITED (IN) 2010-11-11 WO claimed
EP-2427432-A2 NOVEL HETEROCYCLIC COMPOUNDS Torrent Pharmaceuticals Limited (IN) 2012-03-14 EP disclosed
WO-2010128528-A2 NOVEL HETEROCYCLIC COMPOUNDS TORRENT PHARMACEUTICALS LIMITED (IN) 2010-11-11 WO disclosed