SCHEMBL28698477

SCHEMBL28698477

CC(C)(C)OC(=O)N1CCN(c2cc(F)c(CCNC(=O)OCc3ccccc3)cc2F)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.47
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
P2RX7 Q99572 6/20 0.44
SLC2A1 P11166 1/20 0.43
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
ACHE P22303 1/20 0.42
ABCB1 P08183 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
GRM5 P41594 1/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19212145 0.89 GRM5 (0.45) MEN1KMT2AL3MBTL1GRM5ALDH1A1
SCHEMBL28683499 0.88 BACE1 (0.47) BACE1MEN1KMT2AP2RX7SLC2A1
SCHEMBL29576850 0.85 ABCB1 (0.42) MEN1KMT2AKEAP1NFE2L2ABCB1
SCHEMBL21457808 0.85 ABCB1 (0.42) MEN1KMT2AKEAP1NFE2L2ABCB1
SCHEMBL28697404 0.85 ABCB1 (0.43) ABCB1L3MBTL1MAPTSIGMAR1
SCHEMBL29707390 0.85 BACE1 (0.46) BACE1MEN1KMT2AP2RX7SLC2A1
SCHEMBL28673972 0.84 LMNA (0.46) MEN1KMT2AKEAP1NFE2L2L3MBTL1
SCHEMBL29707321 0.82 ABCB1 (0.39) KEAP1NFE2L2ABCB1L3MBTL1LMNA
SCHEMBL21457818 0.82 BACE1 (0.48) BACE1MEN1KMT2AP2RX7SLC2A1
SCHEMBL28697188 0.81 PDK4 (0.45) KEAP1NFE2L2ABCB1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071560-B Thienopyridine carboxamides as ubiquitin-specific protease inhibitors 瓦洛健康公司 2022-01-14 CN disclosed