SCHEMBL28699743

SCHEMBL28699743

COC(=O)CC(N[C@@H]1CCN(C(=O)OC(C)(C)C)C1)c1cccc(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
STS P08842 4/20 0.49
ALDH1A1 P00352 2/20 0.45
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
RAB9A P51151 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
USP30 Q70CQ3 5/20 0.45
MAPK8 P45983 1/20 0.43
AHCY P23526 1/20 0.42
ANO1 Q5XXA6 1/20 0.42
BRD4 O60885 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TP53 P04637 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28686054 0.87 WDR5 (0.42) ALDH1A1
SCHEMBL5575926 0.84 STS (0.57) STSALDH1A1NPC1MAPTMAPK1
SCHEMBL4608693 0.83 STS (0.53) STSALDH1A1NPC1MAPTMAPK1
SCHEMBL28699700 0.82 MAPT (0.41) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL5576153 0.81 STS (0.49) STSALDH1A1NPC1MAPTMAPK1
SCHEMBL5576735 0.80 STS (0.51) STSALDH1A1NPC1MAPTMAPK1
SCHEMBL4608779 0.80 STS (0.49) STSALDH1A1NPC1MAPTMAPK1
SCHEMBL4610832 0.79 STS (0.49) STSALDH1A1NPC1MAPTMAPK1
SCHEMBL4597915 0.79 STS (0.52) STSALDH1A1NPC1MAPTMAPK1
SCHEMBL5573773 0.78 ALDH1A1 (0.49) STSALDH1A1NPC1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354635-B Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2023-04-18 CN disclosed
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed