SCHEMBL28699748

SCHEMBL28699748

COC(=O)C(NC1CCN(CCCc2ccc3c(n2)N(C(=O)O)CCC3)C1)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 8/20 0.35
ITGB6 P18564 4/20 0.35
SIGMAR1 Q99720 1/20 0.35
ITGB3 P05106 4/20 0.35
ITGB5 P18084 3/20 0.35
OPRM1 P35372 1/20 0.34
CHRM3 P20309 1/20 0.34
ITGB1 P05556 2/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
ITGA5 P08648 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28692098 0.83 CCR5 (0.36) ITGAVITGB6
SCHEMBL28690101 0.80 ITGAV (0.37) ITGAVITGB6ITGB3
SCHEMBL28690096 0.80 ITGAV (0.37) ITGAVITGB6ITGB3
SCHEMBL29370436 0.79 ITGAV (0.33) ITGAVITGB6ITGB3ITGB5ITGB1
SCHEMBL28698397 0.78 ITGAV (0.41) ITGAVITGB6ITGB3ITGB5ITGB1
SCHEMBL28708230 0.77 ITGAV (0.40) ITGAVITGB6SIGMAR1ITGB3CHRNB2
SCHEMBL28708228 0.77 ITGAV (0.40) ITGAVITGB6SIGMAR1ITGB3CHRNB2
SCHEMBL28690090 0.77 OPRM1 (0.34) ITGAVITGB6SIGMAR1OPRM1CHRNB2
SCHEMBL28984870 0.76 ITGAV (0.55) ITGAVITGB6ITGB3ITGB5ITGB1
SCHEMBL28709228 0.76 ITGAV (0.55) ITGAVITGB6ITGB3ITGB5ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354635-B Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2023-04-18 CN disclosed
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed