SCHEMBL29370436

SCHEMBL29370436

COC(=O)C(c1ccccc1)N(C)C1[C@H]2CN(CCCc3ccc4c(n3)N(C(=O)O)CCC4)C[C@@H]12

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 9/20 0.33
ITGB3 P05106 5/20 0.33
ITGB5 P18084 3/20 0.33
ITGB1 P05556 1/20 0.33
ITGA5 P08648 1/20 0.33
ITGB6 P18564 4/20 0.32
CCR5 P51681 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28692098 0.89 CCR5 (0.36) ITGAVITGB6CCR5
Trifluoroacetic Acid SCHEMBL29393315 0.80 ITGAV (0.47) ITGAVITGB3ITGB5ITGB1ITGA5
SCHEMBL28708231 0.79 ITGB3 (0.37) ITGAVITGB3ITGB5ITGB1
SCHEMBL28699748 0.79 ITGAV (0.35) ITGAVITGB3ITGB5ITGB1ITGA5
SCHEMBL29369724 0.79 LMNA (0.40) ITGAVITGB3ITGB5ITGB1ITGA5
SCHEMBL28696946 0.79 CCR5 (0.39) ITGAVITGB3ITGB5ITGB6CCR5
SCHEMBL29369797 0.77 HRH3 (0.35) ITGAVITGB3ITGB5ITGB1ITGA5
SCHEMBL29369631 0.77 ITGB3 (0.43) ITGAVITGB3
SCHEMBL29370168 0.75 ITGAV (0.53) ITGAVITGB3ITGB5ITGB1ITGB6
SCHEMBL28337910 0.70 ITGAV (0.40) ITGAVITGB3ITGB5ITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022022364-A1 PYRROLIDINE INTEGRIN MODULATOR AND USE THEREOF 清药同创(北京)药物研发中心有限公司 2022-02-03 WO disclosed