SCHEMBL28700474

SCHEMBL28700474

O=C1NC(=O)c2cc(Br)cc3c(C(F)(F)F)ccc1c23

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.49
PARP1 P09874 2/20 0.37
MEN1 O00255 1/20 0.37
RGS12 O14924 1/20 0.37
USP2 O75604 1/20 0.37
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
MAPT P10636 1/20 0.37
THRB P10828 1/20 0.37
CYP2C9 P11712 1/20 0.37
APEX1 P27695 1/20 0.37
CASP1 P29466 1/20 0.37
BRCA1 P38398 1/20 0.37
MTOR P42345 1/20 0.37
RECQL P46063 1/20 0.37
BLM P54132 1/20 0.37
CASP7 P55210 1/20 0.37
GNAI1 P63096 1/20 0.37
HBB P68871 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1356289 0.79 NPSR1 (0.56) NPSR1PARP1MEN1RGS12USP2
SCHEMBL28261613 0.78 PARP1 (0.57) NPSR1PARP1MEN1RGS12USP2
SCHEMBL4555546 0.68 CES1 (0.56) NPSR1CES1TGM2PARK7
SCHEMBL26644600 0.67 TGM2 (0.46) NPSR1MEN1KMT2ACES1TGM2
SCHEMBL30872149 0.67 TGM2 (0.46) NPSR1MEN1KMT2ACES1TGM2
SCHEMBL7932433 0.66 CES1 (0.42) NPSR1MEN1RGS12POLBCYP3A4
SCHEMBL5749227 0.66 NPSR1 (1.00) NPSR1PARP1MEN1RGS12USP2
SCHEMBL31156926 0.66 NPSR1 (1.00) NPSR1PARP1MEN1RGS12USP2
SCHEMBL383829 0.65 MAOA (0.63) NPSR1PARP1CYP3A4TDP1CES1
SCHEMBL146244 0.64 NPSR1 (0.45) NPSR1PARP1MEN1RGS12USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109053572-B 4-trifluoromethyl-6-bromo-2-substituted acetonitrile-1, 8-naphthalimide compound and preparation method and application thereof 上海应用技术大学 2022-02-11 CN claimed
CN-109053572-B 4-trifluoromethyl-6-bromo-2-substituted acetonitrile-1, 8-naphthalimide compound and preparation method and application thereof 上海应用技术大学 2022-02-11 CN disclosed