SCHEMBL28702102

SCHEMBL28702102

O=C(O)c1ccc2c(=O)n(-c3ccc(OC(F)(F)F)cc3)[nH]c(=O)c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.43
GABRG2 P18507 1/20 0.43
GABRB3 P28472 1/20 0.43
GABRA3 P34903 1/20 0.43
HPD P32754 1/20 0.42
MRGPRX4 Q96LA9 1/20 0.42
AURKA O14965 1/20 0.41
TPX2 Q9ULW0 1/20 0.41
CCNA2 P20248 1/20 0.41
CDK2 P24941 1/20 0.41
CCNA1 P78396 1/20 0.41
EPHX2 P34913 3/20 0.41
FAAH O00519 1/20 0.41
TSHR P16473 1/20 0.40
PDE5A O76074 1/20 0.40
KDM4E B2RXH2 2/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 2/20 0.39
TDP1 Q9NUW8 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20945311 0.95 GABRA1 (0.43) GABRA1GABRG2GABRB3GABRA3HPD
SCHEMBL20945173 0.85 ALDH1A1 (0.46) GABRA1GABRG2GABRB3GABRA3HPD
SCHEMBL20945304 0.81 ALDH1A1 (0.46) GABRA1GABRG2GABRB3GABRA3HPD
SCHEMBL20945293 0.79 TSHR (0.61) GABRA1GABRG2GABRB3GABRA3CCNA2
SCHEMBL20945306 0.77 AR (0.47) GABRA1GABRG2GABRB3GABRA3MRGPRX4
SCHEMBL20945309 0.73 AR (0.47) GABRA1GABRG2GABRB3GABRA3MRGPRX4
SCHEMBL20945265 0.72 GABRA1 (0.44) GABRA1GABRG2GABRB3GABRA3CCNA2
SCHEMBL17826958 0.71 AURKA (0.48) HPDMRGPRX4AURKATPX2EPHX2
SCHEMBL219654 0.71 EPHX2 (0.68) MRGPRX4AURKATPX2EPHX2FAAH
SCHEMBL20945090 0.71 GABRA1 (0.45) GABRA1GABRG2GABRB3GABRA3CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109415345-B Pyridazinone-based broad-spectrum anti-influenza inhibitors 豪夫迈·罗氏有限公司 2022-01-11 CN disclosed