SCHEMBL28704458

SCHEMBL28704458

O=C1C(=O)N(Cc2ccc(Cl)nc2)c2c(Cl)cccc21

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 7/20 0.63
CHRM3 P20309 1/20 0.63
ALDH1A1 P00352 7/20 0.58
ALDH3A1 P30838 5/20 0.58
CES1 P23141 3/20 0.47
TP53 P04637 2/20 0.47
MAPT P10636 2/20 0.47
BCHE P06276 2/20 0.47
ACHE P22303 2/20 0.47
APAF1 O14727 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
ALOX12 P18054 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
CES2 O00748 1/20 0.45
ALDH2 P05091 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29417352 1.00 CHRM5 (0.63) CHRM5CHRM3ALDH1A1ALDH3A1CES1
SCHEMBL28026196 0.83 CHRM5 (0.72) CHRM5CHRM3ALDH1A1ALDH3A1CES1
SCHEMBL30967409 0.82 CHRM5 (0.70) CHRM5CHRM3ALDH1A1ALDH3A1CES1
SCHEMBL770153 0.79 CASP3 (0.54) CHRM5ALDH1A1MAPTCASP3
SCHEMBL30030790 0.77 CHRM5 (1.00) CHRM5CHRM3ALDH1A1ALDH3A1CES1
SCHEMBL22589377 0.73 ALDH3A1 (1.00) ALDH1A1ALDH3A1ALDH2
SCHEMBL12930258 0.73 CHRM5 (0.81) CHRM5CHRM3ALDH1A1ALDH3A1TP53
SCHEMBL22589412 0.73 ALDH1A1 (0.79) ALDH1A1ALDH3A1ALDH2
Bromide SCHEMBL22589442 0.73 ALDH3A1 (1.00) ALDH1A1ALDH3A1ALDH2
SCHEMBL28026197 0.72 CHRM5 (0.61) CHRM5CHRM3ALDH1A1ALDH3A1CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502538-A Substituted 3, 4-dihydroquinazolines for the treatment and prevention of hepatitis B virus infection 豪夫迈·罗氏有限公司 2022-05-13 CN disclosed
CN-114144401-A Novel quinazoline compounds for the treatment and prevention of hepatitis b virus diseases 豪夫迈·罗氏有限公司 2022-03-04 CN disclosed