SCHEMBL28707178

SCHEMBL28707178

CC(=O)Nc1cccc(-c2ccc(-c3nc(C(=O)O)cs3)cc2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.57
SMN1; SMN2 Q16637 7/20 0.57
ALDH1A1 P00352 6/20 0.57
KDM4E B2RXH2 6/20 0.57
MEN1 O00255 4/20 0.57
KMT2A Q03164 4/20 0.57
GAA P10253 2/20 0.57
LMNA P02545 2/20 0.57
HPGD P15428 1/20 0.57
ATM Q13315 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
TDP1 Q9NUW8 1/20 0.55
CYP17A1 P05093 1/20 0.53
CYP11B1 P15538 1/20 0.53
CYP11B2 P19099 1/20 0.53
HTT P42858 2/20 0.52
MAPK1 P28482 1/20 0.52
TP53 P04637 1/20 0.52
NR1H4 Q96RI1 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28701609 0.89 MAPT (0.53) MAPTSMN1; SMN2ALDH1A1KDM4EMEN1
SCHEMBL28720669 0.87 SMN1; SMN2 (0.51) MAPTSMN1; SMN2ALDH1A1KDM4EMEN1
SCHEMBL29654116 0.87 ACHE (0.56) MAPTSMN1; SMN2ALDH1A1KDM4EMEN1
SCHEMBL28707179 0.87 ACHE (0.56) MAPTSMN1; SMN2ALDH1A1KDM4EMEN1
SCHEMBL4444299 0.80 MAPT (0.49) MAPTSMN1; SMN2ALDH1A1HPGDL3MBTL1
SCHEMBL26319518 0.80 ALDH1A1 (0.73) MAPTSMN1; SMN2ALDH1A1KDM4EATM
SCHEMBL25362033 0.78 ALDH1A1 (0.51) MAPTSMN1; SMN2ALDH1A1KDM4EMEN1
SCHEMBL30528155 0.78 ALDH1A1 (0.51) MAPTSMN1; SMN2ALDH1A1KDM4EMEN1
SCHEMBL10068462 0.78 ADRB2 (0.57) MAPTSMN1; SMN2ALDH1A1KDM4EMEN1
SCHEMBL10037335 0.78 ALDH1A1 (0.51) MAPTSMN1; SMN2ALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114249702-A N-aryl- [2,4 '-bithiazole ] -2' -amine compound and preparation and application thereof 沈阳药科大学 2022-03-29 CN disclosed