SCHEMBL28720669

SCHEMBL28720669

CC(=O)Nc1cccc(-c2ccc(-c3nc(C(N)=S)cs3)cc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 8/20 0.51
MAPT P10636 8/20 0.51
ALDH1A1 P00352 5/20 0.51
KDM4E B2RXH2 5/20 0.51
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
GAA P10253 2/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
LMNA P02545 1/20 0.51
HPGD P15428 1/20 0.51
ATM Q13315 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
CYP17A1 P05093 1/20 0.50
CYP11B1 P15538 1/20 0.50
CYP11B2 P19099 1/20 0.50
TDP1 Q9NUW8 1/20 0.49
PARP1 P09874 1/20 0.47
DHODH Q02127 1/20 0.47
MAPK1 P28482 2/20 0.47
HTT P42858 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28701609 0.91 MAPT (0.53) SMN1; SMN2MAPTALDH1A1KDM4EMEN1
SCHEMBL28720671 0.88 SMN1; SMN2 (0.48) SMN1; SMN2MAPTALDH1A1KDM4EMEN1
SCHEMBL29654064 0.88 SMN1; SMN2 (0.48) SMN1; SMN2MAPTALDH1A1KDM4EMEN1
SCHEMBL28707178 0.87 MAPT (0.57) SMN1; SMN2MAPTALDH1A1KDM4EMEN1
SCHEMBL28701610 0.78 ACHE (0.57) SMN1; SMN2MAPTALDH1A1KDM4EMEN1
SCHEMBL29654116 0.74 ACHE (0.56) SMN1; SMN2MAPTALDH1A1KDM4EMEN1
SCHEMBL28707179 0.74 ACHE (0.56) SMN1; SMN2MAPTALDH1A1KDM4EMEN1
SCHEMBL8577619 0.72 SMN1; SMN2 (0.70) SMN1; SMN2ALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL4654909 0.72 ALDH1A1 (0.67) SMN1; SMN2ALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL10663620 0.72 CYP17A1 (0.76) SMN1; SMN2MAPTALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114249702-B N-aryl- [2,4 '-dithiazole ] -2' -amine compound and preparation and application thereof 沈阳药科大学 2023-09-05 CN disclosed
CN-114249702-A N-aryl- [2,4 '-bithiazole ] -2' -amine compound and preparation and application thereof 沈阳药科大学 2022-03-29 CN disclosed