SCHEMBL28708142

SCHEMBL28708142

CC(C)(C)c1ccc(CC(=O)Nc2ccc(=O)n(-c3ccccc3)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.52
NR1H4 Q96RI1 3/20 0.47
PPARG P37231 1/20 0.47
ALDH1A1 P00352 5/20 0.46
RORC P51449 3/20 0.45
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
EPHX2 P34913 1/20 0.43
FLT3 P36888 1/20 0.43
MAPT P10636 3/20 0.43
HPGD P15428 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
RAB9A P51151 2/20 0.43
PKM P14618 1/20 0.43
XBP1 P17861 1/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
CCR6 P51684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28700602 0.89 NLRP3 (0.53) NLRP3RORCSMN1; SMN2EPHX2MAPT
SCHEMBL28698365 0.87 ALDH1A1 (0.52) NLRP3ALDH1A1BCHEACHESMN1; SMN2
SCHEMBL28684550 0.85 MEN1 (0.61) ALDH1A1RORCSMN1; SMN2EPHX2MAPT
SCHEMBL28933313 0.84 MEN1 (0.54) NLRP3ALDH1A1SMN1; SMN2EPHX2MAPT
SCHEMBL28933319 0.84 EPHX2 (0.47) NR1H4ALDH1A1RORCBCHEACHE
SCHEMBL28684557 0.84 ALDH1A1 (0.57) NLRP3ALDH1A1SMN1; SMN2EPHX2MAPT
SCHEMBL28704857 0.84 GAA (0.58) ALDH1A1SMN1; SMN2EPHX2MAPTHPGD
SCHEMBL28691395 0.84 ALDH1A1 (0.64) NLRP3ALDH1A1SMN1; SMN2MAPTHPGD
SCHEMBL28708144 0.82 RAB9A (0.66) NLRP3ALDH1A1SMN1; SMN2MAPTHPGD
SCHEMBL28685814 0.81 KMT2A (0.56) ALDH1A1SMN1; SMN2MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114057630-B Pirfenidone derivative and synthetic method and application thereof 郑州大学 2023-06-02 CN claimed
CN-114057630-A Pirfenidone derivative and synthetic method and application thereof 郑州大学 2022-02-18 CN claimed
CN-114057630-B Pirfenidone derivative and synthetic method and application thereof 郑州大学 2023-06-02 CN disclosed
CN-114057630-A Pirfenidone derivative and synthetic method and application thereof 郑州大学 2022-02-18 CN disclosed