SCHEMBL287119

SCHEMBL287119

O=C(NNC(=O)NC1=CN=CC(CC(=O)c2cccs2)C1)NC1=CN=CC(CC(=O)c2cccs2)C1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.39
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
POLB P06746 2/20 0.39
LMNA P02545 1/20 0.39
ERCC5 P28715 1/20 0.38
FEN1 P39748 1/20 0.38
HPGD P15428 2/20 0.38
GSK3B P49841 1/20 0.38
L3MBTL1 Q9Y468 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MAPT P10636 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
HDAC1 Q13547 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL287370 0.78 ALDH1A1 (0.43) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL287467 0.69 POLB (0.36) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL287683 0.69 NPC1 (0.39) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL287968 0.68 TDP1 (0.41) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL12262036 0.65 ALDH1A1 (0.60) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL662732 0.64 HTT (0.42) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL711360 0.63 RAB9A (0.75) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL5046549 0.62 ALDH1A1 (0.57) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL2966649 0.61 ALDH1A1 (0.64) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL2216212 0.60 ALDH1A1 (1.00) ALDH1A1NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427432-A2 NOVEL HETEROCYCLIC COMPOUNDS Torrent Pharmaceuticals Limited (IN) 2012-03-14 EP disclosed
WO-2010128528-A2 NOVEL HETEROCYCLIC COMPOUNDS TORRENT PHARMACEUTICALS LIMITED (IN) 2010-11-11 WO disclosed