SCHEMBL287370

SCHEMBL287370

O=C(O)C1=CN=CC(CC(=O)c2cccs2)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.43
POLB P06746 4/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 2/20 0.43
DAO P14920 1/20 0.41
ERCC5 P28715 1/20 0.41
FEN1 P39748 1/20 0.41
GSK3B P49841 1/20 0.41
HPGD P15428 5/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
PKM P14618 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL287467 0.79 POLB (0.36) ALDH1A1POLBNPC1RAB9AMEN1
SCHEMBL287683 0.79 NPC1 (0.39) ALDH1A1POLBNPC1RAB9AMEN1
SCHEMBL287119 0.78 ALDH1A1 (0.39) ALDH1A1POLBNPC1RAB9AMEN1
SCHEMBL287825 0.74 ALDH1A1 (0.34) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL287968 0.74 TDP1 (0.41) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL285705 0.73 ALDH1A1 (0.33) ALDH1A1POLBMEN1KMT2ALMNA
SCHEMBL12262036 0.68 ALDH1A1 (0.60) ALDH1A1POLBNPC1RAB9AMEN1
SCHEMBL287432 0.67 TSHR (0.41) ALDH1A1POLBNPC1RAB9AMEN1
SCHEMBL5046549 0.65 ALDH1A1 (0.57) ALDH1A1POLBNPC1RAB9AMEN1
SCHEMBL287282 0.65 TDP1 (0.43) ALDH1A1NPC1RAB9AKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427432-A2 NOVEL HETEROCYCLIC COMPOUNDS Torrent Pharmaceuticals Limited (IN) 2012-03-14 EP disclosed
WO-2010128528-A2 NOVEL HETEROCYCLIC COMPOUNDS TORRENT PHARMACEUTICALS LIMITED (IN) 2010-11-11 WO disclosed