SCHEMBL28720200

SCHEMBL28720200

c1ccc(-c2ccccc2CNCCc2c[nH]cn2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 1/20 0.45
HDAC3 O15379 3/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC2 Q92769 3/20 0.40
HDAC6 Q9UBN7 3/20 0.40
HDAC4 P56524 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
TACR1 P25103 1/20 0.39
CD274 Q9NZQ7 3/20 0.39
ITGB1 P05556 2/20 0.37
ITGA4 P13612 2/20 0.37
ITGB7 P26010 2/20 0.37
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4605920 0.80 GAA (0.53) MPO
SCHEMBL2103787 0.78 DPP4 (0.43) HDAC3HDAC1HDAC2HDAC6CD274
SCHEMBL17654953 0.76 EPHX2 (0.33)
SCHEMBL6180571 0.75 SIGMAR1 (0.50)
SCHEMBL28930178 0.75 MPO (0.62) SCN8AHDAC3HDAC1HDAC2HDAC6
SCHEMBL10478067 0.74 EPHX2 (0.54) MPO
SCHEMBL31364605 0.74 ALDH1A1 (0.31)
SCHEMBL31364603 0.74 ALDH1A1 (0.31)
SCHEMBL10045086 0.71 SCN8A (0.61) SCN8AHDAC3HDAC1HDAC2HDAC6
SCHEMBL10045151 0.70 SCN8A (0.60) SCN8AHDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109305942-B Preparation method and application of 4-imidazolyl-containing glutaminyl cyclase inhibitor 深圳大学 2022-04-22 CN disclosed
CN-108912051-B Glutaminyl cyclase inhibitor containing 4-imidazolyl 深圳大学 2022-04-15 CN disclosed