SCHEMBL28720236

SCHEMBL28720236

COc1cccc(SC(F)(F)/C(F)=C/CN2C(=O)c3ccccc3C2=O)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.42
HTR1A P08908 4/20 0.41
GAA P10253 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
MMP2 P08253 1/20 0.39
MMP9 P14780 1/20 0.39
NPC1 O15118 1/20 0.38
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
HTT P42858 1/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37
MAPK1 P28482 1/20 0.37
ATM Q13315 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28720240 1.00 RAB9A (0.42) RAB9AHTR1AGAARXFP1MEN1
SCHEMBL29486879 1.00 RAB9A (0.42) RAB9AHTR1AGAARXFP1MEN1
SCHEMBL28703606 0.84 CASP3 (0.42) RAB9AMEN1ALDH1A1KMT2ANPC1
SCHEMBL22918281 0.84 CASP3 (0.42) RAB9AMEN1ALDH1A1KMT2ANPC1
SCHEMBL29486855 0.84 CASP3 (0.42) RAB9AMEN1ALDH1A1KMT2ANPC1
SCHEMBL28713856 0.81 PKM (0.39) RAB9AMEN1ALDH1A1MAPTKMT2A
SCHEMBL22918300 0.81 PKM (0.39) RAB9AMEN1ALDH1A1MAPTKMT2A
SCHEMBL29486871 0.81 PKM (0.39) RAB9AMEN1ALDH1A1MAPTKMT2A
SCHEMBL22918403 0.79 HTR1A (0.43) RAB9AHTR1AGAAMEN1ALDH1A1
SCHEMBL29852306 0.77 CASP3 (0.35) RAB9AGAAMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114286816-A Difluoro-halogenated allylamine sulfone derivative inhibitor of lysyl oxidase, preparation method and application thereof 法玛西斯有限公司 2022-04-05 CN disclosed