SCHEMBL28724743

SCHEMBL28724743

N#Cc1c(C(F)(F)F)n[nH]c1-c1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.43
MAPT P10636 3/20 0.43
KDM4E B2RXH2 3/20 0.43
HTT P42858 2/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 2/20 0.43
ERBB2 P04626 1/20 0.41
HSD17B10 Q99714 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 2/20 0.39
NCOA1 Q15788 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
DHODH Q02127 1/20 0.38
MEN1 O00255 1/20 0.38
ADORA1 P30542 2/20 0.38
MAPK14 Q16539 4/20 0.37
GCGR P47871 2/20 0.37
MAPK13 O15264 1/20 0.37
ALOX5 P09917 1/20 0.37
MAPK12 P53778 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28724777 0.88 MAPT (0.41) KMT2AMAPTKDM4EHTTALDH1A1
SCHEMBL28724773 0.88 KIF11 (0.46) KMT2AMAPTKDM4EALDH1A1HSD17B10
SCHEMBL28724765 0.88 KIF11 (0.46) DHODHMAPK14GCGRMAPK13ALOX5
SCHEMBL28724776 0.86 GRM5 (0.44) KMT2AMAPTKDM4EHTTALDH1A1
SCHEMBL28724775 0.86 GRM5 (0.44) KMT2AMAPTKDM4EALDH1A1GAA
SCHEMBL28724767 0.86 GAA (0.44) KMT2AMAPTHTTALDH1A1GAA
SCHEMBL28724772 0.84 DHODH (0.43) KMT2AMAPTKDM4EHTTALDH1A1
SCHEMBL28724967 0.82 MAPT (0.47) KMT2AMAPTKDM4EALDH1A1MEN1
SCHEMBL28724763 0.80 ABCC8 (0.47) KMT2AMAPTALDH1A1LMNADHODH
SCHEMBL29483457 0.80 IKBKB (0.43) KMT2AKDM4EHTTALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114349703-B Trifluoromethyl-4-cyano pyrazole compound, and preparation method and application thereof 天津大学 2024-05-10 CN disclosed
CN-114349703-A Trifluoromethyl-4-cyanopyrazole compound, and preparation method and application thereof 天津大学 2022-04-15 CN disclosed