SCHEMBL28724765

SCHEMBL28724765

N#Cc1ccc(-c2[nH]nc(C(F)(F)F)c2C#N)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.46
DGAT1 O75907 1/20 0.40
SOAT1 P35610 1/20 0.40
KCNH2 Q12809 1/20 0.40
GYS1 P13807 1/20 0.40
TRPA1 O75762 1/20 0.39
SCN5A Q14524 1/20 0.39
SCN9A Q15858 1/20 0.39
NOTUM Q6P988 1/20 0.39
CYP11B2 P19099 1/20 0.38
MAPK14 Q16539 3/20 0.37
MAPK13 O15264 2/20 0.37
MAPK12 P53778 2/20 0.37
MAPK11 Q15759 2/20 0.37
GCGR P47871 2/20 0.37
ALOX5 P09917 1/20 0.37
DHODH Q02127 1/20 0.36
PTPN5 P54829 1/20 0.36
RAF1 P04049 1/20 0.35
MMP3 P08254 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28724773 0.88 KIF11 (0.46) KIF11DGAT1SOAT1KCNH2NOTUM
SCHEMBL28724743 0.88 KMT2A (0.43) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL28724777 0.88 MAPT (0.41) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL28724767 0.86 GAA (0.44) DHODH
SCHEMBL28724775 0.86 GRM5 (0.44) KIF11
SCHEMBL28724776 0.86 GRM5 (0.44)
SCHEMBL28724772 0.84 DHODH (0.43) KIF11NOTUMDHODH
SCHEMBL28724967 0.82 MAPT (0.47)
SCHEMBL28724763 0.80 ABCC8 (0.47) GYS1NOTUMMAPK14MAPK13MAPK12
SCHEMBL28724771 0.80 IKBKB (0.43) GYS1NOTUMMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114349703-B Trifluoromethyl-4-cyano pyrazole compound, and preparation method and application thereof 天津大学 2024-05-10 CN disclosed
CN-114349703-A Trifluoromethyl-4-cyanopyrazole compound, and preparation method and application thereof 天津大学 2022-04-15 CN disclosed